1. From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors. Issue 13 (1st July 2017) Authors: Liang, Jun; Labadie, Sharada; Zhang, Birong; Ortwine, Daniel F.; Patel, Snahel; Vinogradova, Maia; Kiefer, James R.; Mauer, Till; Gehling, Victor S.; Harmange, Jean-Christophe; Cummings, Richard; Lai, Tommy; Liao, Jiangpeng; Zheng, Xiaoping; Liu, Yichin; Gustafson, Amy; Van der Porten, Erica; Mao... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 13(2017) Page Start: 2974 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Lead optimization of a pyrazolo[1, 5-a]pyrimidin-7(4H)-one scaffold to identify potent, selective and orally bioavailable KDM5 inhibitors suitable for in vivo biological studies. Issue 16 (15th August 2016) Authors: Liang, Jun; Zhang, Birong; Labadie, Sharada; Ortwine, Daniel F.; Vinogradova, Maia; Kiefer, James R.; Gehling, Victor S.; Harmange, Jean-Christophe; Cummings, Richard; Lai, Tommy; Liao, Jiangpeng; Zheng, Xiaoping; Liu, Yichin; Gustafson, Amy; Van der Porten, Erica; Mao, Weifeng; Liederer, Bianca ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 16(2016) Page Start: 4036 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗