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Author/Creator Tokarski, John

1. Development of BET inhibitors as potential treatments for cancer: A new carboline chemotype. (1st November 2021)

Authors:
Hill, Matthew D.; Quesnelle, Claude; Tokarski, John; Fang, Haiquan; Fanslau, Carolynn; Haarhoff, Zuzana; Kramer, Melissa; Madari, Shilpa; Wiebesiek, Amy; Morrison, John; Simmermacher-Mayer, Jean; Sinz, Michael; Westhouse, Richard; Xie, Chunshan; Zhao, Jiuqiao; Huang, Lisa; Sheriff, Steven; Yan, C...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 51(2021)
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Journal Article
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2. Development of BET inhibitors as potential treatments for cancer: A search for structural diversity. (15th July 2021)

Authors:
Hill, Matthew D.; Fang, Haiquan; Tokarski, John; Fanslau, Carolynn; Haarhoff, Zuzana; Huang, Christine; Kramer, Melissa; Menard, Krista; Monereau, Laura; Morrison, John; Ranasinghe, Asoka; Shields, Eric E.; Tye, Ching Kim; Westhouse, Richard; Everlof, Gerry; Sheriff, Steven; Yan, Chunhong; Marsil...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 44(2021)
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Journal Article
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3. Discovery of highly potent, selective, covalent inhibitors of JAK3. Issue 20 (15th October 2017)

Authors:
Kempson, James; Ovalle, Damaso; Guo, Junqing; Wrobleski, Stephen T.; Lin, Shuqun; Spergel, Steven H.; Duan, James J.-W.; Jiang, Bin; Lu, Zhonghui; Das, Jagabandhu; Yang, Bingwei V.; Hynes, John; Wu, Hong; Tokarski, John; Sack, John S.; Khan, Javed; Schieven, Gary; Blatt, Yuval; Chaudhry, Charu; S...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 20(2017)
Page Start:
4622
Record Type:
Journal Article
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4. The discovery of BMS-737 as a potent, CYP17 lyase-selective inhibitor for the treatment of castration-resistant prostate cancer. (1st November 2022)

Authors:
Padmakar Darne, Chetan; Velaparthi, Upender; Saulnier, Mark; Frennesson, David; Liu, Peiying; Huang, Audris; Tokarski, John; Fura, Aberra; Spires, Thomas; Newitt, John; Spires, Vanessa M.; Obermeier, Mary T.; Elzinga, Paul A.; Gottardis, Marco M.; Jayaraman, Lata; Vite, Gregory D.; Balog, Aaron
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 75(2022)
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Record Type:
Journal Article
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