1. A small molecule inhibitor of PCSK9 that antagonizes LDL receptor binding via interaction with a cryptic PCSK9 binding groove. Issue 6 (15th March 2020) Authors: Evison, Benny J.; Palmer, James T.; Lambert, Gilles; Treutlein, Herbert; Zeng, Jun; Nativel, Brice; Chemello, Kévin; Zhu, Qing; Wang, Jie; Teng, Yanfen; Tang, Wei; Xu, Yanfeng; Rathi, Anuj Kumar; Kumar, Sanjay; Suchowerska, Alexandra K.; Parmar, Jasneet; Dixon, Ian; Kelly, Graham E.; Bonnar, James Journal: Bioorganic & medicinal chemistry Issue: Volume 28:Issue 6(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗