1. A PEGylated analog of short-length Neuromedin U with potent anorectic and anti-obesity effects. Issue 8 (15th April 2017) Authors: Inooka, Hiroshi; Sakamoto, Kotaro; Shinohara, Tokuyuki; Masuda, Yasushi; Terada, Michiko; Kumano, Satoshi; Yokoyama, Kotaro; Noguchi, Jiro; Nishizawa, Naoki; Kamiguchi, Hidenori; Fujita, Hisashi; Asami, Taiji; Takekawa, Shiro; Ohtaki, Tetsuya Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 8(2017) Page Start: 2307 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. A potent and selective natriuretic peptide receptor-3 blocker 11-mer peptide created by hybridization of musclin and atrial natriuretic peptide. Issue 15 (1st August 2017) Authors: Nishizawa, Naoki; Nakamura, Goshi; Noguchi, Yoko; Nakagawa, Hideyuki; Shimizu, Ayako; Nakayama, Masaharu; Takekawa, Shiro; Asami, Taiji Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 15(2017) Page Start: 3542 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. A potent neuromedin U receptor 2-selective alkylated peptide. Issue 20 (15th October 2017) Authors: Nishizawa, Naoki; Kanematsu-Yamaki, Yoko; Funata, Masaaki; Nagai, Hiroaki; Shimizu, Ayako; Fujita, Hisashi; Sakamoto, Junichi; Takekawa, Shiro; Asami, Taiji Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 20(2017) Page Start: 4626 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Antiobesity and emetic effects of a short-length peptide YY analog and its PEGylated and alkylated derivatives. Issue 3 (1st February 2018) Authors: Niida, Ayumu; Kanematsu-Yamaki, Yoko; Asakawa, Tomoko; Ishimura, Yoshimasa; Fujita, Hisashi; Matsumiya, Kouta; Nishizawa, Naoki; Adachi, Yusuke; Mochida, Taisuke; Tsuchimori, Kazue; Yoneyama-Hirozane, Mariko; Sakamoto, Junichi; Hirabayashi, Hideki; Fukui, Hideo; Takekawa, Shiro; Asami, Taiji Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 3(2018) Page Start: 566 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Differential effects of selective agonists of neuromedin U1 and U2 receptors in obese and diabetic mice. (18th December 2017) Authors: Nagai, Hiroaki; Kaisho, Tomoko; Yokoyama, Kotaro; Asakawa, Tomoko; Fujita, Hisashi; Matsumiya, Kouta; Noguchi, Jiro; Tsuchimori, Kazue; Nishizawa, Naoki; Kanematsu‐Yamaki, Yoko; Dote, Katsuko; Inooka, Hiroshi; Sakamoto, Jun‐ichi; Ohtaki, Tetsuya; Asami, Taiji; Takekawa, Shiro Journal: British journal of pharmacology Issue: Volume 175:Number 2(2018) Page Start: 359 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Highly potent antiobesity effect of a short-length peptide YY analog in mice. Issue 20 (15th October 2017) Authors: Nishizawa, Naoki; Niida, Ayumu; Adachi, Yusuke; Kanematsu-Yamaki, Yoko; Masuda, Yasushi; Kumano, Satoshi; Yokoyama, Kotaro; Noguchi, Yoko; Asakawa, Tomoko; Hirabayashi, Hideki; Amano, Nobuyuki; Takekawa, Shiro; Ohtaki, Tetsuya; Asami, Taiji Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 20(2017) Page Start: 5718 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Identification and Characterization of a New Series of Ghrelin O-Acyl Transferase Inhibitors. (February 2018) Authors: Yoneyama-Hirozane, Mariko; Deguchi, Kohei; Hirakawa, Takeshi; Ishii, Tsuyoshi; Odani, Tomoyuki; Matsui, Junji; Nakano, Yoshihide; Imahashi, Kenichi; Takakura, Nobuyuki; Chisaki, Ikumi; Takekawa, Shiro; Sakamoto, Junichi Journal: SLAS discovery Issue: Volume 23:Number 2(2018) Page Start: 154 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Inhibition of MGAT2 modulates fat‐induced gut peptide release and fat intake in normal mice and ameliorates obesity and diabetes in ob/ob mice fed on a high‐fat diet. Issue 3 (5th February 2020) Authors: Mochida, Taisuke; Take, Kazumi; Maki, Toshiyuki; Nakakariya, Masanori; Adachi, Ryutaro; Sato, Kenjiro; Kitazaki, Tomoyuki; Takekawa, Shiro Journal: FEBS open bio Issue: Volume 10:Issue 3(2020) Page Start: 316 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Optimization of a novel series of N-phenylindoline-5-sulfonamide-based acyl CoA:monoacylglycerol acyltransferase-2 inhibitors: Mitigation of CYP3A4 time-dependent inhibition and phototoxic liabilities. Issue 15 (1st August 2015) Authors: Sato, Kenjiro; Takahagi, Hiroki; Kubo, Osamu; Hidaka, Kousuke; Yoshikawa, Takeshi; Kamaura, Masahiro; Nakakariya, Masanori; Amano, Nobuyuki; Adachi, Ryutaro; Maki, Toshiyuki; Take, Kazumi; Takekawa, Shiro; Kitazaki, Tomoyuki; Maekawa, Tsuyoshi Journal: Bioorganic & medicinal chemistry Issue: Volume 23:Issue 15(2015) Page Start: 4544 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Potent antiobesity effect of a short-length peptide YY-analogue continuously administered in mice. Issue 16 (15th August 2017) Authors: Nishizawa, Naoki; Niida, Ayumu; Adachi, Yusuke; Masuda, Yasushi; Kumano, Satoshi; Yokoyama, Kotaro; Asakawa, Tomoko; Hirabayashi, Hideki; Amano, Nobuyuki; Takekawa, Shiro; Ohtaki, Tetsuya; Asami, Taiji Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 16(2017) Page Start: 3829 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗