1. Discovery of MDV6058 (PF-06952229), a selective and potent TGFβR1 inhibitor: Design, synthesis and optimization. (1st November 2022) Authors: Pujala, Brahmam; Ramachandran, Sreekanth A.; Sonawane, Mukesh; Kamble, Maruti M.; Panpatil, Dayanand; Adhikari, Swati; Soni, Sanjeev; Subbareddy, Venkata; Shinde, Bharat U.; Nayak, Anjan K.; Bansal, Chandni; Gupta, Ashu; Mukherjee, Kakoli; Agarwal, Anil K.; Guerrero, Javier; Herrera, Francisco J.... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 75(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗