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Author/Creator Stefanski, Kevin

1. Discovery and SAR of pyrrolo[2, 1-f][1, 2, 4]triazin-4-amines as potent and selective PI3Kδ inhibitors. Issue 17 (1st September 2016)

Authors:
Bhide, Rajeev S.; Neels, James; Qin, Lan-Ying; Ruan, Zheming; Stachura, Sylwia; Weigelt, Carolyn; Sack, John S.; Stefanski, Kevin; Gu, Xiaomei; Xie, Jenny H.; Goldstine, Christine B.; Skala, Stacey; Pedicord, Donna L.; Ruepp, Stefan; Dhar, T.G. Murali; Carter, Percy H.; Salter-Cid, Luisa M.; Poss...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 17(2016)
Page Start:
4256
Record Type:
Journal Article
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2. Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2, 1-f][1, 2, 4]triazin-4-amine derivatives as highly potent and selective PI3Kδ inhibitors. Issue 4 (15th February 2017)

Authors:
Qin, Lan-Ying; Ruan, Zheming; Cherney, Robert J.; Dhar, T.G. Murali; Neels, James; Weigelt, Carolyn A.; Sack, John S.; Srivastava, Anurag S.; Cornelius, Lyndon A.M.; Tino, Joseph A.; Stefanski, Kevin; Gu, Xiaomei; Xie, Jenny; Susulic, Vojkan; Yang, Xiaoxia; Yarde-Chinn, Melissa; Skala, Stacey; Bo...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 4(2017)
Page Start:
855
Record Type:
Journal Article
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3. Oral Delivery of Highly Lipophilic Poorly Water‐Soluble Drugs: Spray‐Dried Dispersions to Improve Oral Absorption and Enable High‐Dose Toxicology Studies of a P2Y1 Antagonist. Issue 12 (10th October 2014)

Authors:
Chen, Xue‐Qing; Stefanski, Kevin; Shen, Hong; Huang, Christine; Caporuscio, Christian; Yang, Wu; Lam, Patrick; Su, Ching; Gudmundsson, Olafur; Hageman, Michael
Journal:
Journal of pharmaceutical sciences
Issue:
Volume 103:Issue 12(2014:Dec.)
Page Start:
3924
Record Type:
Journal Article
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4. Tricyclic sulfones as potent, selective and efficacious RORγt inverse agonists – Exploring C6 and C8 SAR using late-stage functionalization. Issue 23 (1st December 2020)

Authors:
Shi, Qing; Xiao, Zili; Yang, Michael G.; Marcoux, David; Cherney, Robert J.; Yip, Shiuhang; Li, Peng; Wu, Dauh-Rurng; Weigelt, Carolyn A.; Sack, John; Khan, Javed; Ruzanov, Max; Wang, Jinhong; Yarde, Melissa; Ellen Cvijic, Mary; Li, Sha; Shuster, David J.; Xie, Jenny; Sherry, Tara; Obermeier, Mary
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 23(2020)
Page Start:
Record Type:
Journal Article
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5. Ultrasensitive quantitative LC–MS/MS of an inhibitor of apoptosis protein's antagonist in plasma using protein target affinity extraction. (February 2016)

Authors:
Discenza, Lorell N; Cornelius, Georgia; Gan, Jinping; Szapiel, Nicolas; Talbott, Randy L; Chaudhry, Charu; Roy, Anirban; Borzilleri, Robert M; Vuppugalla, Ragini; Stefanski, Kevin; Moore, Robin; D'Arienzo, Celia J; Olah, Timothy V; Mehl, John T
Journal:
Bioanalysis
Issue:
Volume 8:Number 4(2016)
Page Start:
265
Record Type:
Journal Article
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