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- Steadman, David [remove] 7
- Pharmaceutical chemistry -- Periodicals 4
- 572 3
- Biochemistry -- Periodicals 2
- Bioorganic chemistry -- Periodicals 2
- 005.8 1
- 615.19 1
- 615.19005 1
- 616.9041 1
- Alzheimer's disease -- Neurodegeneration -- Neuroinflammation -- Drug discovery pipeline -- Symptomatic treatments -- Disease modification 1
- Aβ amyloid-beta -- AD Alzheimer's disease -- ADME absorption distribution metabolism elimination -- CNS central nervous system -- ER efflux ratio -- FP fluorophosphonate -- HBD hydrogen bond donor -- MLM mouse liver microsomes -- MPO multiparameter optimization -- OPTS trisodium 8-octanoyloxypyrene-1, 3, 6-trisulfonate -- P-gp P-glycoprotein -- SAR structure activity relationship -- SBDD structure based drug design -- TPSA topological polar surface area -- UPLC–MS ultra performance liquid chromatography–mass spectrometer -- HBTU O-(1H-Benzotriazol-1-yl)-N, N, N′, N′-tetra-methyluronium hexafluorophosphate 1