1. MARK inhibitors: Declaring a No-Go decision on a chemical series based on extensive DMPK experimentation. Issue 1 (1st January 2017) Authors: Haidle, Andrew M.; Childers, Kaleen K.; Zabierek, Anna A.; Katz, Jason D.; Jewell, James P.; Hou, Yongquan; Altman, Michael D.; Szewczak, Alexander; Chen, Dapeng; Harsch, Andreas; Hayashi, Mansuo; Warren, Lee; Hutton, Michael; Nuthall, Hugh; Stanton, Matt G.; Davies, Ian W.; Munoz, Ben; Northrup,... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 1(2017) Page Start: 109 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Structure guided design of a series of selective pyrrolopyrimidinone MARK inhibitors. Issue 1 (1st January 2017) Authors: Katz, Jason D.; Haidle, Andrew; Childers, Kaleen K.; Zabierek, Anna A.; Jewell, James P.; Hou, Yongquan; Altman, Michael D.; Szewczak, Alexander; Chen, Dapeng; Harsch, Andreas; Hayashi, Mansuo; Warren, Lee; Hutton, Michael; Nuthall, Hugh; Su, Hua-Poo; Munshi, Sanjeev; Stanton, Matt G.; Davies, Ia... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 1(2017) Page Start: 114 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗