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Author/Creator Snell, Gyorgy

1. Discovery and optimization of 1, 7-disubstituted-2, 2-dimethyl-2, 3-dihydroquinazolin-4(1H)-ones as potent and selective PKCθ inhibitors. Issue 11 (1st June 2016)

Authors:
Katoh, Taisuke; Takai, Takafumi; Yukawa, Takafumi; Tsukamoto, Tetsuya; Watanabe, Etsurou; Mototani, Hideyuki; Arita, Takeo; Hayashi, Hiroki; Nakagawa, Hideyuki; Klein, Michael G.; Zou, Hua; Sang, Bi-Ching; Snell, Gyorgy; Nakada, Yoshihisa
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 24:Issue 11(2016)
Page Start:
2466
Record Type:
Journal Article
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2. Discovery of a novel B-cell lymphoma 6 (BCL6)–corepressor interaction inhibitor by utilizing structure-based drug design. Issue 17 (1st September 2017)

Authors:
Yasui, Takeshi; Yamamoto, Takeshi; Sakai, Nozomu; Asano, Kouhei; Takai, Takafumi; Yoshitomi, Yayoi; Davis, Melinda; Takagi, Terufumi; Sakamoto, Kotaro; Sogabe, Satoshi; Kamada, Yusuke; Lane, Weston; Snell, Gyorgy; Iwata, Masashi; Goto, Masayuki; Inooka, Hiroshi; Sakamoto, Jun-ichi; Nakada, Yoshih...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 25:Issue 17(2017)
Page Start:
4876
Record Type:
Journal Article
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3. Discovery of benzimidazole derivatives as orally active renin inhibitors: Optimization of 3, 5-disubstituted piperidine to improve pharmacokinetic profile. Issue 12 (23rd July 2018)

Authors:
Tokuhara, Hidekazu; Imaeda, Yasuhiro; Fukase, Yoshiyuki; Iwanaga, Koichi; Taya, Naohiro; Watanabe, Koji; Kanagawa, Ray; Matsuda, Keisuke; Kajimoto, Yumiko; Kusumoto, Keiji; Kondo, Mitsuyo; Snell, Gyorgy; Behnke, Craig A.; Kuroita, Takanobu
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 26:Issue 12(2018)
Page Start:
3261
Record Type:
Journal Article
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4. Novel approach of fragment-based lead discovery applied to renin inhibitors. Issue 22 (15th November 2016)

Authors:
Tawada, Michiko; Suzuki, Shinkichi; Imaeda, Yasuhiro; Oki, Hideyuki; Snell, Gyorgy; Behnke, Craig A.; Kondo, Mitsuyo; Tarui, Naoki; Tanaka, Toshimasa; Kuroita, Takanobu; Tomimoto, Masaki
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 24:Issue 22(2016)
Page Start:
6066
Record Type:
Journal Article
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5. Novel approach of fragment-based lead discovery applied to renin inhibitors. Issue 22 (15th November 2016)

Authors:
Tawada, Michiko; Suzuki, Shinkichi; Imaeda, Yasuhiro; Oki, Hideyuki; Snell, Gyorgy; Behnke, Craig A.; Kondo, Mitsuyo; Tarui, Naoki; Tanaka, Toshimasa; Kuroita, Takanobu; Tomimoto, Masaki
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 24:Issue 22(2016)
Page Start:
6066
Record Type:
Journal Article
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7. Structure-based design of a new series of N-(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors. Issue 22 (15th November 2016)

Authors:
Imaeda, Yasuhiro; Tawada, Michiko; Suzuki, Shinkichi; Tomimoto, Masaki; Kondo, Mitsuyo; Tarui, Naoki; Sanada, Tsukasa; Kanagawa, Ray; Snell, Gyorgy; Behnke, Craig A.; Kubo, Keiji; Kuroita, Takanobu
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 24:Issue 22(2016)
Page Start:
5771
Record Type:
Journal Article
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8. Structure-based design of a new series of N-(piperidin-3-yl)pyrimidine-5-carboxamides as renin inhibitors. Issue 22 (15th November 2016)

Authors:
Imaeda, Yasuhiro; Tawada, Michiko; Suzuki, Shinkichi; Tomimoto, Masaki; Kondo, Mitsuyo; Tarui, Naoki; Sanada, Tsukasa; Kanagawa, Ray; Snell, Gyorgy; Behnke, Craig A.; Kubo, Keiji; Kuroita, Takanobu
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 24:Issue 22(2016)
Page Start:
5771
Record Type:
Journal Article
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9. Structure-based design, synthesis, and biological evaluation of imidazo[1, 2-b]pyridazine-based p38 MAP kinase inhibitors. Issue 3 (1st February 2018)

Authors:
Kaieda, Akira; Takahashi, Masashi; Takai, Takafumi; Goto, Masayuki; Miyazaki, Takahiro; Hori, Yuri; Unno, Satoko; Kawamoto, Tomohiro; Tanaka, Toshimasa; Itono, Sachiko; Takagi, Terufumi; Hamada, Teruki; Shirasaki, Mikio; Okada, Kengo; Snell, Gyorgy; Bragstad, Ken; Sang, Bi-Ching; Uchikawa, Osamu;...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 26:Issue 3(2018)
Page Start:
647
Record Type:
Journal Article
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10. Structure‐Based Design, Synthesis, and Biological Evaluation of Imidazo[4, 5‐b]pyridin‐2‐one‐Based p38 MAP Kinase Inhibitors: Part 1. (18th April 2019)

Authors:
Kaieda, Akira; Takahashi, Masashi; Fukuda, Hiromi; Okamoto, Rei; Morimoto, Shinji; Gotoh, Masayuki; Miyazaki, Takahiro; Hori, Yuri; Unno, Satoko; Kawamoto, Tomohiro; Tanaka, Toshimasa; Itono, Sachiko; Takagi, Terufumi; Sugimoto, Hiroshi; Okada, Kengo; Snell, Gyorgy; Bertsch, Ryan; Nguyen, Jasmine...
Journal:
ChemMedChem
Issue:
Volume 14:Number 10(2019)
Page Start:
1022
Record Type:
Journal Article
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