1. Discovery and SAR of pyrrolo[2, 1-f][1, 2, 4]triazin-4-amines as potent and selective PI3Kδ inhibitors. Issue 17 (1st September 2016) Authors: Bhide, Rajeev S.; Neels, James; Qin, Lan-Ying; Ruan, Zheming; Stachura, Sylwia; Weigelt, Carolyn; Sack, John S.; Stefanski, Kevin; Gu, Xiaomei; Xie, Jenny H.; Goldstine, Christine B.; Skala, Stacey; Pedicord, Donna L.; Ruepp, Stefan; Dhar, T.G. Murali; Carter, Percy H.; Salter-Cid, Luisa M.; Poss... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 17(2016) Page Start: 4256 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2, 1-f][1, 2, 4]triazin-4-amine derivatives as highly potent and selective PI3Kδ inhibitors. Issue 4 (15th February 2017) Authors: Qin, Lan-Ying; Ruan, Zheming; Cherney, Robert J.; Dhar, T.G. Murali; Neels, James; Weigelt, Carolyn A.; Sack, John S.; Srivastava, Anurag S.; Cornelius, Lyndon A.M.; Tino, Joseph A.; Stefanski, Kevin; Gu, Xiaomei; Xie, Jenny; Susulic, Vojkan; Yang, Xiaoxia; Yarde-Chinn, Melissa; Skala, Stacey; Bo... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 4(2017) Page Start: 855 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗