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Author/Creator Siemeister, Gerhard

2. Back Cover: Modular Assembly of Allosteric MEK Inhibitor Structural Elements Unravels Potency and Feedback‐Modulation Handles (ChemMedChem 12/2015). Issue 12 (December 2015)

Authors:
Hartung, Ingo V.; Pühler, Florian; Neuhaus, Roland; Scholz, Arne; Siemeister, Gerhard; Geisler, Jens; Hillig, Roman C.; von Ahsen, Oliver; Hitchcock, Marion
Journal:
ChemMedChem
Issue:
Volume 10:Issue 12(2015:Dec.)
Page Start:
2116
Record Type:
Journal Article
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3. Cover Picture: The Lab Oddity Prevails: Discovery of Pan‐CDK Inhibitor (R)‐S‐Cyclopropyl‐S‐(4‐{[4‐{[(1R, 2R)‐2‐hydroxy‐1‐methylpropyl]oxy}‐5‐(trifluoromethyl)pyrimidin‐2‐yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer (ChemMedChem 7/2013). Issue 7 (26th June 2013)

Authors:
Lücking, Ulrich; Jautelat, Rolf; Krüger, Martin; Brumby, Thomas; Lienau, Philip; Schäfer, Martina; Briem, Hans; Schulze, Julia; Hillisch, Alexander; Reichel, Andreas; Wengner, Antje Margret; Siemeister, Gerhard
Journal:
ChemMedChem
Issue:
Volume 8:Issue 7(2013:Jul.)
Page Start:
1021
Record Type:
Journal Article
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4. Identification of Atuveciclib (BAY 1143572), the First Highly Selective, Clinical PTEFb/CDK9 Inhibitor for the Treatment of Cancer. (16th October 2017)

Authors:
Lücking, Ulrich; Scholz, Arne; Lienau, Philip; Siemeister, Gerhard; Kosemund, Dirk; Bohlmann, Rolf; Briem, Hans; Terebesi, Ildiko; Meyer, Kirstin; Prelle, Katja; Denner, Karsten; Bömer, Ulf; Schäfer, Martina; Eis, Knut; Valencia, Ray; Ince, Stuart; von Nussbaum, Franz; Mumberg, Dominik; Ziegelbau...
Journal:
ChemMedChem
Issue:
Volume 12:Number 21(2017)
Page Start:
1776
Record Type:
Journal Article
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5. Modular Assembly of Allosteric MEK Inhibitor Structural Elements Unravels Potency and Feedback‐Modulation Handles. Issue 12 (6th November 2015)

Authors:
Hartung, Ingo V.; Pühler, Florian; Neuhaus, Roland; Scholz, Arne; Siemeister, Gerhard; Geisler, Jens; Hillig, Roman C.; von Ahsen, Oliver; Hitchcock, Marion
Journal:
ChemMedChem
Issue:
Volume 10:Issue 12(2015:Dec.)
Page Start:
2004
Record Type:
Journal Article
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6. Optimization of allosteric MEK inhibitors. Part 2: Taming the sulfamide group balances compound distribution properties. Issue 1 (1st January 2016)

Authors:
Hartung, Ingo V.; Hammer, Stefanie; Hitchcock, Marion; Neuhaus, Roland; Scholz, Arne; Siemeister, Gerhard; Bohlmann, Rolf; Hillig, Roman C.; Pühler, Florian
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 1(2016)
Page Start:
186
Record Type:
Journal Article
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7. The Lab Oddity Prevails: Discovery of Pan‐CDK Inhibitor (R)‐S‐Cyclopropyl‐S‐(4‐{[4‐{[(1R, 2R)‐2‐hydroxy‐1‐methylpropyl]oxy}‐5‐(trifluoromethyl)pyrimidin‐2‐yl]amino}phenyl)sulfoximide (BAY 1000394) for the Treatment of Cancer. Issue 7 (13th May 2013)

Authors:
Lücking, Ulrich; Jautelat, Rolf; Krüger, Martin; Brumby, Thomas; Lienau, Philip; Schäfer, Martina; Briem, Hans; Schulze, Julia; Hillisch, Alexander; Reichel, Andreas; Wengner, Antje Margret; Siemeister, Gerhard
Journal:
ChemMedChem
Issue:
Volume 8:Issue 7(2013:Jul.)
Page Start:
1067
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗