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Author/Creator Sherer, Brian

1. Optimization of the efflux ratio and permeability of covalent irreversible BTK inhibitors. Issue 20 (1st November 2018)

Authors:
Qiu, Hui; Liu-Bujalski, Lesley; Caldwell, Richard D.; Viacava Follis, Ariele; Gardberg, Anna; Goutopoulos, Andreas; Grenningloh, Roland; Head, Jared; Johnson, Theresa; Jones, Christopher C.V.; Jones, Reinaldo; Mochalkin, Igor; Morandi, Federica; Neagu, Constantin; Potnick, Justin; Sherer, Brian
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 20(2018)
Page Start:
3307
Record Type:
Journal Article
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2. Discovery of 4-aminopyrimidine analogs as highly potent dual P70S6K/Akt inhibitors. (15th October 2021)

Authors:
Xiao, Yufang; Huck, Bayard R.; Lan, Ruoxi; DeSelm, Lizbeth; Chen, Xiaoling; Qiu, Hui; Neagu, Constantin; Johnson, Theresa; Mochalkin, Igor; Gardberg, Anna; Jiang, Xuliang; Tian, Hui; Dutt, Vikram; Santos, Dusica; Head, Jared; Jackson, Jennifer; Syed, Sakeena; Lin, Jing; Wilker, Erik; Ma, Jianguo
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 50(2021)
Page Start:
Record Type:
Journal Article
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3. O37 M5049, a novel potent and selective inhibitor of toll-like receptors 7 and 8 (TLR 7/8). (23rd March 2020)

Authors:
Sherer, Brian; Bender, Andrew T; Pereira, Albertina; Reissig, Sonja; Haselmayer, Philipp; Okitsu, Shinji L; Tzvetkov, Evgeni; Przetak, Melinda; Morse, Noune Tahmassian; Vlach, Jaromir
Journal:
Lupus science & medicine
Issue:
Volume 7(2020)Supplement 1
Page Start:
A28
Record Type:
Journal Article
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4. Corrigendum to "Discovery of 4-aminopyrimidine analogs as highly potent dual P70S6K/Akt inhibitors" [Bioorgan. Med. Chem. Lett. 50 (2021) 128352]. (1st July 2022)

Authors:
Xiao, Yufang; Huck, Bayard R.; Lan, Ruoxi; DeSelm, Lizbeth; Chen, Xiaoling; Qiu, Hui; Neagu, Constantin; Johnson, Theresa; Mochalkin, Igor; Gardberg, Anna; Jiang, Xuliang; Tian, Hui; Dutt, Vikram; Santos, Dusica; Head, Jared; Jackson, Jennifer; Syed, Sakeena; Lin, Jing; Wilker, Erik; Ma, Jianguo
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 67(2022)
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Record Type:
Journal Article
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5. Discovery of potent, highly selective covalent irreversible BTK inhibitors from a fragment hit. Issue 17 (15th September 2018)

Authors:
Qiu, Hui; Liu-Bujalski, Lesley; Caldwell, Richard D; Follis, Ariele Viacava; Gardberg, Anna; Goutopoulos, Andreas; Grenningloh, Roland; Head, Jared; Johnson, Theresa; Jones, Reinaldo; Mochalkin, Igor; Morandi, Federica; Neagu, Constantin; Sherer, Brian
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 17(2018)
Page Start:
2939
Record Type:
Journal Article
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6. Synthesis and SAR development of quinoline analogs as novel P2X7 receptor antagonists. Issue 13 (1st July 2019)

Authors:
Xiao, Yufang; Karra, Srinivasa; Goutopoulos, Andreas; Morse, Noune Tahmassian; Zhang, Susan; Dhanabal, Mohanraj; Tian, Hui; Seenisamy, Jeyaprakashnarayanan; Jayadevan, Jayashankaran; Caldwell, Richard; Potnick, Justin; Bleich, Matthew; Chekler, Eugene; Sherer, Brian; Sriraman, Venkataraman
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 29:Issue 13(2019)
Page Start:
1660
Record Type:
Journal Article
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7. Discovery of potent and selective reversible Bruton's tyrosine kinase inhibitors. (15th June 2021)

Authors:
Qiu, Hui; Ali, Zahid; Bender, Andrew; Caldwell, Richard; Chen, Yi-Ying; Fang, Zhizhou; Gardberg, Anna; Glaser, Nina; Goettsche, Anja; Goutopoulos, Andreas; Grenningloh, Roland; Hanschke, Bettina; Head, Jared; Johnson, Theresa; Jones, Christopher; Jones, Reinaldo; Kulkarni, Shashank; Maurer, Chris...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 40(2021)
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Record Type:
Journal Article
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8. Discovery of a novel series of pyridine and pyrimidine carboxamides as potent and selective covalent inhibitors of Btk. Issue 21 (15th November 2018)

Authors:
Caldwell, Richard; Liu-Bujalski, Lesley; Qiu, Hui; Mochalkin, Igor; Jones, Reinaldo; Neagu, Constantin; Goutopoulos, Andreas; Grenningloh, Roland; Johnson, Theresa; Sherer, Brian; Gardberg, Anna; Follis, Ariele Viacava; Morandi, Federica; Head, Jared
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 21(2018)
Page Start:
3419
Record Type:
Journal Article
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9. Discovery of Affinity‐Based Probes for Btk Occupancy Assays. (9th January 2019)

Authors:
Qiu, Hui; Caldwell, Richard; Liu‐Bujalski, Lesley; Goutopoulos, Andreas; Jones, Reinaldo; Potnick, Justin; Sherer, Brian; Bender, Andrew; Grenningloh, Roland; Xu, Daigen; Gardberg, Anna; Mochalkin, Igor; Johnson, Theresa; Viacava Follis, Ariele; Head, Jared; Morandi, Federica
Journal:
ChemMedChem
Issue:
Volume 14:Number 2(2019)
Page Start:
217
Record Type:
Journal Article
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