1. Increasing metabolic stability via the deuterium kinetic isotope effect: An example from a proline-amide-urea aminothiazole series of phosphatidylinositol-3 kinase alpha inhibitors. Issue 19 (1st October 2016) Authors: Fairhurst, Robin A.; Caravatti, Giorgio; Guagnano, Vito; Aichholz, Reiner; Blanz, Joachim; Blasco, Francesca; Wipfli, Peter; Fritsch, Christine; Maira, Sauveur-Michel; Schnell, Christian; Seiler, Frank H. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 19(2016) Page Start: 4729 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗