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Author/Creator Ruzanov, Max

1. Developing Adnectins That Target SRC Co-Activator Binding to PXR: A Structural Approach toward Understanding Promiscuity of PXR. Issue 4 (27th February 2015)

Authors:
Khan, Javed A.; Camac, Daniel M.; Low, Simon; Tebben, Andrew J.; Wensel, David L.; Wright, Martin C.; Su, Julie; Jenny, Victoria; Gupta, Ruchira Das; Ruzanov, Max; Russo, Katie A.; Bell, Aneka; An, Yongmi; Bryson, James W.; Gao, Mian; Gambhire, Pallavi; Baldwin, Eric T.; Gardner, Daniel; Cavallar...
Journal:
Journal of molecular biology
Issue:
Volume 427:Issue 4(2015:Feb. 15)
Page Start:
924
Record Type:
Journal Article
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2. Discovery of 2, 6–difluorobenzyl ether series of phenyl ((R)–3–phenylpyrrolidin–3–yl)sulfones as surprisingly potent, selective and orally bioavailable RORγt inverse agonists. Issue 19 (1st October 2020)

Authors:
Duan, James J.-W.; Jiang, Bin; Lu, Zhonghui; Stachura, Sylwia; Weigelt, Carolyn A.; Sack, John S.; Khan, Javed; Ruzanov, Max; Wu, Dauh–Rurng; Yarde, Melissa; Shen, Ding–Ren; Zhao, Qihong; Salter–Cid, Luisa M.; Carter, Percy H.; Murali Dhar, T.G.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 19(2020)
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Record Type:
Journal Article
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3. Heterobicyclic inhibitors of transforming growth factor beta receptor I (TGFβRI). Issue 5 (1st March 2018)

Authors:
Harikrishnan, Lalgudi S.; Warrier, Jayakumar; Tebben, Andrew J.; Tonukunuru, Gopikishan; Madduri, Sudhakara R.; Baligar, Vishweshwaraiah; Mannoori, Raju; Seshadri, Balaji; Rahaman, Hasibur; Arunachalam, P.N.; Dikundwar, Amol G.; Fink, Brian E.; Fargnoli, Joseph; Fereshteh, Mark; Fan, Yi; Lippy, J...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 26:Issue 5(2018)
Page Start:
1026
Record Type:
Journal Article
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4. Identification of potent, selective and orally bioavailable phenyl ((R)-3-phenylpyrrolidin-3-yl)sulfone analogues as RORγt inverse agonists. Issue 16 (15th August 2019)

Authors:
Lu, Zhonghui; Duan, James J.-W.; Xiao, Haiyun; Neels, James; Wu, Dauh-Rurng; Weigelt, Carolyn A.; Sack, John S.; Khan, Javed; Ruzanov, Max; An, Yongmi; Yarde, Melissa; Karmakar, Ananta; Vishwakrishnan, Sureshbabu; Baratam, Venkata; Shankarappa, Harisha; Vanteru, Sridhar; Babu, Venkatesh; Basha, M...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 29:Issue 16(2019)
Page Start:
2265
Record Type:
Journal Article
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5. Signal transfer in human protein tyrosine phosphatase PTP1B from allosteric inhibitor P00058. Issue 24 (26th December 2022)

Authors:
Chirgadze, Yuri N.; Battaile, Kevin P.; Likhachev, Ilya V.; Balabaev, Nikolay K.; Gordon, Roni D.; Romanov, Vladimir; Lin, Andres; Karisch, Robert; Lam, Robert; Ruzanov, Max; Brazhnikov, Evgeniy V.; Pai, Emil F.; Neel, Benjamin G.; Chirgadze, Nickolay Y.
Journal:
Journal of biomolecular structure & dynamics
Issue:
Volume 40:Issue 24(2022)
Page Start:
13823
Record Type:
Journal Article
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6. Substituted benzyloxytricyclic compounds as retinoic acid-related orphan receptor gamma t (RORγt) agonists. Issue 12 (15th June 2020)

Authors:
Harikrishnan, Lalgudi S.; Gill, Patrice; Kamau, Muthoni G.; Qin, Lan-Ying; Ruan, Zheming; O'Malley, Daniel; Huynh, Tram; Stachura, Sylwia; Cavallaro, Cullen L.; Lu, Zhonghui; J.-W. Duan, James; Weigelt, Carolyn A.; Sack, John S.; Ruzanov, Max; Khan, Javed; Gururajan, Murali; Wong, Jessica J.; Hua...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 12(2020)
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Journal Article
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7. Substituted diaryl ether compounds as retinoic acid-related orphan Receptor-γt (RORγt) agonists. (1st March 2021)

Authors:
Ruan, Zheming; Park, Peter K.; Wei, Donna; Purandare, Ashok; Wan, Honghe; O'Malley, Daniel; Stachura, Sylwia; Perez, Heidi; Cavallaro, Cullen L.; Weigelt, Carolyn A.; Sack, John S.; Ruzanov, Max; Khan, Javed; Gururajan, Murali; Wong, Jessica J.; Huang, Yanling; Yarde, Melissa; Li, Zhuyin; Chen, C...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 35(2021)
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Record Type:
Journal Article
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8. Tricyclic sulfones as potent, selective and efficacious RORγt inverse agonists – Exploring C6 and C8 SAR using late-stage functionalization. Issue 23 (1st December 2020)

Authors:
Shi, Qing; Xiao, Zili; Yang, Michael G.; Marcoux, David; Cherney, Robert J.; Yip, Shiuhang; Li, Peng; Wu, Dauh-Rurng; Weigelt, Carolyn A.; Sack, John; Khan, Javed; Ruzanov, Max; Wang, Jinhong; Yarde, Melissa; Ellen Cvijic, Mary; Li, Sha; Shuster, David J.; Xie, Jenny; Sherry, Tara; Obermeier, Mary
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 23(2020)
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Journal Article
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9. Using yeast surface display to engineer a soluble and crystallizable construct of hematopoietic progenitor kinase 1 (HPK1). Issue 1 (13th January 2021)

Authors:
Lau, Wai L.; Pearce, Bradley; Malakian, Heather; Rodrigo, Iyoncy; Xie, Dianlin; Gao, Mian; Marsilio, Frank; Chang, Chiehying; Ruzanov, Max; Muckelbauer, Jodi K.; Newitt, John A.; Lipovšek, Daša; Sheriff, Steven
Journal:
Acta crystallographica
Issue:
Volume 77:Issue 1(2021)
Page Start:
22
Record Type:
Journal Article
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