1. Structure-based design of Trifarotene (CD5789), a potent and selective RARγ agonist for the treatment of acne. Issue 10 (1st June 2018) Authors: Thoreau, Etienne; Arlabosse, Jean-Marie; Bouix-Peter, Claire; Chambon, Sandrine; Chantalat, Laurent; Daver, Sébastien; Dumais, Laurence; Duvert, Gwenaëlle; Feret, Angélique; Ouvry, Gilles; Pascau, Jonathan; Raffin, Catherine; Rodeville, Nicolas; Soulet, Catherine; Tabet, Samuel; Talano, Sandrine;... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 10(2018) Page Start: 1736 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. An efficient multi-component synthesis of N-1-alkylated 5-nitrouracils from α-amino acids. Issue 22 (1st June 2016) Authors: Boiteau, Jean-Guy; Bouix-Peter, Claire; Chambon, Sandrine; Clary, Laurence; Daver, Sebastien; Dumais, Laurence; Fournier, Jean-François; Harris, Craig S.; Mebrouk, Kenny; Millois, Corinne; Pierre, Romain; Rodeville, Nicolas; Talano, Sandrine; Tomas, Loïc Journal: Tetrahedron letters Issue: Volume 57:Issue 22(2016) Page Start: 2367 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis. Issue 4 (15th February 2018) Authors: Boiteau, Jean-Guy; Ouvry, Gilles; Arlabosse, Jean-Marie; Astri, Stéphanie; Beillard, Audrey; Bhurruth-Alcor, Yushma; Bonnary, Laetitia; Bouix-Peter, Claire; Bouquet, Karine; Bourotte, Marilyne; Cardinaud, Isabelle; Comino, Catherine; Deprez, Benoît; Duvert, Denis; Féret, Angélique; Hacini-Rachine... Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 4(2018) Page Start: 945 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗