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Author/Creator Rai, Roopa

1. Targeting prostate cancer with compounds possessing dual activity as androgen receptor antagonists and HDAC6 inhibitors. Issue 21 (1st November 2016)

Authors:
Jadhavar, Pradeep S.; Ramachandran, Sreekanth A.; Riquelme, Eduardo; Gupta, Ashu; Quinn, Kevin P.; Shivakumar, Devleena; Ray, Soumya; Zende, Dnyaneshwar; Nayak, Anjan K.; Miglani, Sandeep K.; Sathe, Balaji D.; Raja, Mohd.; Farias, Olivia; Alfaro, Ivan; Belmar, Sebastián; Guerrero, Javier; Bernale...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 21(2016)
Page Start:
5222
Record Type:
Journal Article
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2. Discovery of MDV6058 (PF-06952229), a selective and potent TGFβR1 inhibitor: Design, synthesis and optimization. (1st November 2022)

Authors:
Pujala, Brahmam; Ramachandran, Sreekanth A.; Sonawane, Mukesh; Kamble, Maruti M.; Panpatil, Dayanand; Adhikari, Swati; Soni, Sanjeev; Subbareddy, Venkata; Shinde, Bharat U.; Nayak, Anjan K.; Bansal, Chandni; Gupta, Ashu; Mukherjee, Kakoli; Agarwal, Anil K.; Guerrero, Javier; Herrera, Francisco J....
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 75(2022)
Page Start:
Record Type:
Journal Article
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3. Discovery of pyrazolopyrimidine derivatives as novel inhibitors of ataxia telangiectasia and rad3 related protein (ATR). Issue 4 (15th February 2017)

Authors:
Ramachandran, Sreekanth A.; Jadhavar, Pradeep S.; Singh, Manvendra P.; Sharma, Ankesh; Bagle, Gaurav N.; Quinn, Kevin P.; Wong, Po-yin; Protter, Andrew A.; Rai, Roopa; Pham, Son M.; Lindquist, Jeffrey N.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 4(2017)
Page Start:
750
Record Type:
Journal Article
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4. Novel 3-methylindoline inhibitors of EZH2: Design, synthesis and SAR. Issue 2 (15th January 2017)

Authors:
Ansari, Amantullah; Satalkar, Sharad; Patil, Varshavekumar; Shete, Amit S.; Kaur, Simranjeet; Gupta, Ashu; Singh, Siddhartha; Raja, Mohd.; Severance, Daniel L.; Bernales, Sebastián; Chakravarty, Sarvajit; Hung, David T.; Pham, Son M.; Herrera, Francisco J.; Rai, Roopa
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 2(2017)
Page Start:
217
Record Type:
Journal Article
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5. Design, synthesis and optimization of bis-amide derivatives as CSF1R inhibitors. Issue 10 (15th May 2017)

Authors:
Ramachandran, Sreekanth A.; Jadhavar, Pradeep S.; Miglani, Sandeep K.; Singh, Manvendra P.; Kalane, Deepak P.; Agarwal, Anil K.; Sathe, Balaji D.; Mukherjee, Kakoli; Gupta, Ashu; Haldar, Srijan; Raja, Mohd; Singh, Siddhartha; Pham, Son M.; Chakravarty, Sarvajit; Quinn, Kevin; Belmar, Sebastian; A...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 10(2017)
Page Start:
2153
Record Type:
Journal Article
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6. Temozolomide analogs with improved brain/plasma ratios – Exploring the possibility of enhancing the therapeutic index of temozolomide. Issue 20 (15th October 2016)

Authors:
Rai, Roopa; Banerjee, Monali; Wong, Darren H.; McCullagh, Emma; Gupta, Ashu; Tripathi, Shailendra; Riquelme, Eduardo; Jangir, Ramnivas; Yadav, Shyamraj; Raja, Mohd.; Melkani, Pankaj; Dixit, Vikas; Patil, Umesh; Shrivastava, Ritesh; Middya, Sandip; Olivares, Felipe; Guerrero, Javier; Surya, Arjun;...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 20(2016)
Page Start:
5103
Record Type:
Journal Article
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