1. Development of isoquinolinone derivatives as immunoproteasome inhibitors. (1st January 2022) Authors: Ettari, Roberta; Iraci, Nunzio; Di Chio, Carla; Previti, Santo; Danzè, Mariafernanda; Zappalà, Maria Journal: Bioorganic & medicinal chemistry letters Issue: Volume 55(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Development of novel 1, 4-benzodiazepine-based Michael acceptors as antitrypanosomal agents. Issue 15 (1st August 2016) Authors: Ettari, Roberta; Previti, Santo; Cosconati, Sandro; Maiorana, Santina; Schirmeister, Tanja; Grasso, Silvana; Zappalà, Maria Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 15(2016) Page Start: 3453 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Development of Novel Benzodiazepine‐Based Peptidomimetics as Inhibitors of Rhodesain from Trypanosoma brucei rhodesiense. (5th May 2020) Authors: Di Chio, Carla; Previti, Santo; Amendola, Giorgio; Cosconati, Sandro; Schirmeister, Tanja; Zappalà, Maria; Ettari, Roberta Journal: ChemMedChem Issue: Volume 15:Number 11(2020) Page Start: 995 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Development of novel dipeptide-like rhodesain inhibitors containing the 3-bromoisoxazoline warhead in a constrained conformation. Issue 21 (1st November 2015) Authors: Ettari, Roberta; Pinto, Andrea; Previti, Santo; Tamborini, Lucia; Angelo, Ilenia C.; La Pietra, Valeria; Marinelli, Luciana; Novellino, Ettore; Schirmeister, Tanja; Zappalà, Maria; Grasso, Silvana; De Micheli, Carlo; Conti, Paola Journal: Bioorganic & medicinal chemistry Issue: Volume 23:Issue 21(2015) Page Start: 7053 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Drug combination studies of curcumin and genistein against rhodesain of Trypanosoma brucei rhodesiense. Issue 24 (17th December 2019) Authors: Ettari, Roberta; Previti, Santo; Maiorana, Santina; Allegra, Alessandro; Schirmeister, Tanja; Grasso, Silvana; Zappalà, Maria Journal: Natural product research Issue: Volume 33:Issue 24(2019) Page Start: 3577 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Drug combination studies of PS-1 and quercetin against rhodesain of Trypanosoma brucei rhodesiense. Issue 16 (29th July 2022) Authors: Di Chio, Carla; Previti, Santo; De Luca, Fabiola; Allegra, Alessandro; Zappalà, Maria; Ettari, Roberta Journal: Natural product research Issue: Volume 36:Issue 16(2022) Page Start: 4282 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Evaluation of curcumin irreversibility. Issue 22 (16th November 2020) Authors: Ettari, Roberta; Previti, Santo; Maiorana, Santina; Allegra, Alessandro; Schirmeister, Tanja; Grasso, Silvana; Zappalà, Maria Journal: Natural product research Issue: Volume 34:Issue 22(2020) Page Start: 3159 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Identification of 2-thioxoimidazolidin-4-one derivatives as novel noncovalent proteasome and immunoproteasome inhibitors. Issue 3 (1st February 2018) Authors: Maccari, Rosanna; Ettari, Roberta; Adornato, Ilenia; Naß, Alexandra; Wolber, Gerhard; Bitto, Alessandra; Mannino, Federica; Aliquò, Federica; Bruno, Giuseppe; Nicolò, Francesco; Previti, Santo; Grasso, Silvana; Zappalà, Maria; Ottanà, Rosaria Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 3(2018) Page Start: 278 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Peptidyl Vinyl Ketone Irreversible Inhibitors of Rhodesain: Modifications of the P2 Fragment. (7th July 2020) Authors: Maiorana, Santina; Ettari, Roberta; Previti, Santo; Amendola, Giorgio; Wagner, Annika; Cosconati, Sandro; Hellmich, Ute A.; Schirmeister, Tanja; Zappalà, Maria Journal: ChemMedChem Issue: Volume 15:Number 16(2020) Page Start: 1552 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Synthesis and biological evaluation of novel peptidomimetics as rhodesain inhibitors. (1st November 2016) Authors: Ettari, Roberta; Previti, Santo; Cosconati, Sandro; Kesselring, Jochen; Schirmeister, Tanja; Grasso, Silvana; Zappalà, Maria Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 31:Number 6(2016:Dec.) Page Start: 1184 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗