1. A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced‐Fit Pocket Stabilized by a Cation–π Interaction1. (12th May 2014) Authors: Rooney, Timothy P. C.; Filippakopoulos, Panagis; Fedorov, Oleg; Picaud, Sarah; Cortopassi, Wilian A.; Hay, Duncan A.; Martin, Sarah; Tumber, Anthony; Rogers, Catherine M.; Philpott, Martin; Wang, Minghua; Thompson, Amber L.; Heightman, Tom D.; Pryde, David C.; Cook, Andrew; Paton, Robert S.; Müll... Journal: Angewandte Chemie Issue: Volume 126:Number 24(2014) Page Start: 6240 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. A Series of Potent CREBBP Bromodomain Ligands Reveals an Induced‐Fit Pocket Stabilized by a Cation–π Interaction1. Issue 24 (12th May 2014) Authors: Rooney, Timothy P. C.; Filippakopoulos, Panagis; Fedorov, Oleg; Picaud, Sarah; Cortopassi, Wilian A.; Hay, Duncan A.; Martin, Sarah; Tumber, Anthony; Rogers, Catherine M.; Philpott, Martin; Wang, Minghua; Thompson, Amber L.; Heightman, Tom D.; Pryde, David C.; Cook, Andrew; Paton, Robert S.; Müll... Journal: Angewandte Chemie international edition Issue: Volume 53:Issue 24(2014) Page Start: 6126 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. BET bromodomain ligands: Probing the WPF shelf to improve BRD4 bromodomain affinity and metabolic stability. Issue 11 (15th July 2018) Authors: Jennings, Laura E.; Schiedel, Matthias; Hewings, David S.; Picaud, Sarah; Laurin, Corentine M.C.; Bruno, Paul A.; Bluck, Joseph P.; Scorah, Amy R.; See, Larissa; Reynolds, Jessica K.; Moroglu, Mustafa; Mistry, Ishna N.; Hicks, Amy; Guzanov, Pavel; Clayton, James; Evans, Charles N.G.; Stazi, Giuli... Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 11(2018) Page Start: 2937 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery of Benzo[d]imidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain. (15th September 2022) Authors: Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca Journal: ChemMedChem Issue: Volume 17:Number 20(2022) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Evaluation of linker length effects on a BET bromodomain probe. Issue 68 (6th August 2019) Authors: Traquete, Rui; Henderson, Elizabeth; Picaud, Sarah; Cal, Pedro M. S. D.; Sieglitz, Florian; Rodrigues, Tiago; Oliveira, Rudi; Filippakopoulos, Panagis; Bernardes, Gonçalo J. L. Journal: Chemical communications Issue: Volume 55:Issue 68(2019) Page Start: 10128 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Front Cover: Discovery of Benzo[d]imidazole‐6‐sulfonamides as Bromodomain and Extra‐Terminal Domain (BET) Inhibitors with Selectivity for the First Bromodomain (ChemMedChem 20/2022). (19th October 2022) Authors: Cipriano, Alessandra; Milite, Ciro; Feoli, Alessandra; Viviano, Monica; Pepe, Giacomo; Campiglia, Pietro; Sarno, Giuliana; Picaud, Sarah; Imaide, Satomi; Makukhin, Nikolai; Filippakopoulos, Panagis; Ciulli, Alessio; Castellano, Sabrina; Sbardella, Gianluca Journal: ChemMedChem Issue: Volume 17:Number 20(2022) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Identification of a PGXPP degron motif in dishevelled and structural basis for its binding to the E3 ligase KLHL12. Issue 6 (24th June 2020) Authors: Chen, Zhuoyao; Wasney, Gregory A.; Picaud, Sarah; Filippakopoulos, Panagis; Vedadi, Masoud; D'Angiolella, Vincenzo; Bullock, Alex N. Journal: Open biology Issue: Volume 10:Issue 6(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Probing BRD Inhibition Substituent Effects in Bulky Analogues of (+)‐JQ1. Issue 3 (3rd February 2021) Authors: Hassell‐Hart, Storm; Picaud, Sarah; Lengacher, Raphael; Csucker, Joshua; Millet, Regis; Gasser, Gilles; Alberto, Roger; Maple, Hannah; Felix, Robert; Leśnikowski, Zbigniew J.; Stewart, Helen J. S.; Chevassut, Timothy J.; Morley, Simon; Filippakopoulos, Panagis; Spencer, John Journal: Helvetica chimica acta Issue: Volume 104:Issue 3(2021) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Small molecule inhibitors reveal an indispensable scaffolding role of RIPK2 in NOD2 signaling. (19th July 2018) Authors: Hrdinka, Matous; Schlicher, Lisa; Dai, Bing; Pinkas, Daniel M; Bufton, Joshua C; Picaud, Sarah; Ward, Jennifer A; Rogers, Catherine; Suebsuwong, Chalada; Nikhar, Sameer; Cuny, Gregory D; Huber, Kilian VM; Filippakopoulos, Panagis; Bullock, Alex N; Degterev, Alexei; Gyrd‐Hansen, Mads Journal: EMBO journal Issue: Volume 37:Number 17(2018) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗