1. Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis. (6th February 2018) Authors: Ouvry, Gilles; Atrux‐Tallau, Nicolas; Bihl, Franck; Bondu, Aline; Bouix‐Peter, Claire; Carlavan, Isabelle; Christin, Olivier; Cuadrado, Marie‐Josée; Defoin‐Platel, Claire; Deret, Sophie; Duvert, Denis; Feret, Christophe; Forissier, Mathieu; Fournier, Jean‐François; Froude, David; Hacini‐Rachinel,... Journal: ChemMedChem Issue: Volume 13:Number 4(2018) Page Start: 321 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis. Issue 4 (15th February 2018) Authors: Boiteau, Jean-Guy; Ouvry, Gilles; Arlabosse, Jean-Marie; Astri, Stéphanie; Beillard, Audrey; Bhurruth-Alcor, Yushma; Bonnary, Laetitia; Bouix-Peter, Claire; Bouquet, Karine; Bourotte, Marilyne; Cardinaud, Isabelle; Comino, Catherine; Deprez, Benoît; Duvert, Denis; Féret, Angélique; Hacini-Rachine... Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 4(2018) Page Start: 945 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists. Issue 23 (1st December 2016) Authors: Ouvry, Gilles; Bouix-Peter, Claire; Ciesielski, Fabrice; Chantalat, Laurent; Christin, Olivier; Comino, Catherine; Duvert, Denis; Feret, Christophe; Harris, Craig S.; Lamy, Laurent; Luzy, Anne-Pascale; Musicki, Branislav; Orfila, Danielle; Pascau, Jonathan; Parnet, Véronique; Perrin, Agnès; Pierr... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 23(2016) Page Start: 5802 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Identification of novel TACE inhibitors compatible with topical application. Issue 8 (15th April 2017) Authors: Ouvry, Gilles; Berton, Yaël; Bhurruth-Alcor, Yushma; Bonnary, Laetitia; Bouix-Peter, Claire; Bouquet, Karine; Bourotte, Marilyne; Chambon, Sandrine; Comino, Catherine; Deprez, Benoît; Duvert, Denis; Duvert, Gwenaëlle; Hacini-Rachinel, Feriel; Harris, Craig S.; Luzy, Anne-Pascale; Mathieu, Arnaud;... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 8(2017) Page Start: 1848 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. New Caspase-1 inhibitor by scaffold hopping into bio-inspired 3D-fragment space. Issue 24 (15th December 2017) Authors: Brethon, Anne; Chantalat, Laurent; Christin, Olivier; Clary, Laurence; Fournier, Jean-François; Gastreich, Marcus; Harris, Craig S.; Isabet, Tatiana; Pascau, Jonathan; Thoreau, Etienne; Roche, Didier; Rodeschini, Vincent Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 24(2017) Page Start: 5373 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Squaramides as novel class I and IIB histone deacetylase inhibitors for topical treatment of cutaneous t-cell lymphoma. Issue 17 (15th September 2018) Authors: Fournier, Jean-François; Bhurruth-Alcor, Yushma; Musicki, Branislav; Aubert, Jérome; Aurelly, Michèle; Bouix-Peter, Claire; Bouquet, Karinne; Chantalat, Laurent; Delorme, Marion; Drean, Bénédicte; Duvert, Gwenaelle; Fleury-Bregeot, Nicolas; Gauthier, Blanche; Grisendi, Karine; Harris, Craig S.; H... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 17(2018) Page Start: 2985 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Structure-based design of Trifarotene (CD5789), a potent and selective RARγ agonist for the treatment of acne. Issue 10 (1st June 2018) Authors: Thoreau, Etienne; Arlabosse, Jean-Marie; Bouix-Peter, Claire; Chambon, Sandrine; Chantalat, Laurent; Daver, Sébastien; Dumais, Laurence; Duvert, Gwenaëlle; Feret, Angélique; Ouvry, Gilles; Pascau, Jonathan; Raffin, Catherine; Rodeville, Nicolas; Soulet, Catherine; Tabet, Samuel; Talano, Sandrine;... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 10(2018) Page Start: 1736 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Sulfoximines as potent RORγ inverse agonists. Issue 8 (1st May 2018) Authors: Ouvry, Gilles; Bihl, Franck; Bouix-Peter, Claire; Christin, Olivier; Defoin-Platel, Claire; Deret, Sophie; Feret, Christophe; Froude, David; Hacini-Rachinel, Feriel; Harris, Craig S.; Hervouet, Catherine; Lafitte, Guillaume; Luzy, Anne-Pascale; Musicki, Branislav; Orfila, Danielle; Parnet, Veroni... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 8(2018) Page Start: 1269 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗