1. Design, synthesis, and evaluation of novel N-1 fluoroquinolone derivatives: Probing for binding contact with the active site tyrosine of gyrase. Issue 10 (1st June 2018) Authors: Towle, Tyrell R.; Kulkarni, Chaitanya A.; Oppegard, Lisa M.; Williams, Bridget P.; Picha, Taylor A.; Hiasa, Hiroshi; Kerns, Robert J. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 10(2018) Page Start: 1903 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Suppression of gyrase-mediated resistance by C7 aryl fluoroquinolones. Issue 7 (16th March 2016) Authors: Malik, Muhammad; Mustaev, Arkady; Schwanz, Heidi A.; Luan, Gan; Shah, Nirali; Oppegard, Lisa M.; de Souza, Ernane C.; Hiasa, Hiroshi; Zhao, Xilin; Kerns, Robert J.; Drlica, Karl Journal: Nucleic acids research Issue: Volume 44:Issue 7(2016) Page Start: 3304 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗