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Author/Creator Musil, Djordje

1. Discovery of potent and selective CDK8 inhibitors from an HSP90 pharmacophore. Issue 5 (1st March 2016)

Authors:
Schiemann, Kai; Mallinger, Aurélie; Wienke, Dirk; Esdar, Christina; Poeschke, Oliver; Busch, Michael; Rohdich, Felix; Eccles, Suzanne A.; Schneider, Richard; Raynaud, Florence I.; Czodrowski, Paul; Musil, Djordje; Schwarz, Daniel; Urbahns, Klaus; Blagg, Julian
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 5(2016)
Page Start:
1443
Record Type:
Journal Article
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2. Identification and characterization of M6903, an antagonistic anti–TIM-3 monoclonal antibody. (1st January 2020)

Authors:
Zhang, Dong; Jiang, Feng; Zaynagetdinov, Rinat; Huang, Hui; Sood, Vanita D.; Wang, Hong; Zhao, Xinyan; Jenkins, Molly H.; Ji, Qingyong; Wang, Youbin; Nannemann, David P.; Musil, Djordje; Wesolowski, John; Paoletti, Andrea; Bartholomew, Tin; Derner, Melissa G.; An, Qi; Iffland, Christel; Halle, Jo...
Journal:
Oncoimmunology
Issue:
Volume 9:Number 1(2020)
Page Start:
Record Type:
Journal Article
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3. Ligand‐Induced Conformational Changes in HSP90 Monitored Time Resolved and Label Free—Towards a Conformational Activity Screening for Drug Discovery. Issue 31 (3rd July 2018)

Authors:
Güldenhaupt, Jörn; Amaral, Marta; Kötting, Carsten; Schartner, Jonas; Musil, Djordje; Frech, Matthias; Gerwert, Klaus
Journal:
Angewandte Chemie international edition
Issue:
Volume 57:Issue 31(2018)
Page Start:
9955
Record Type:
Journal Article
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4. Novel reversible methionine aminopeptidase-2 (MetAP-2) inhibitors based on purine and related bicyclic templates. Issue 3 (1st February 2017)

Authors:
Heinrich, Timo; Buchstaller, Hans-Peter; Cezanne, Bertram; Rohdich, Felix; Bomke, Jörg; Friese-Hamim, Manja; Krier, Mireille; Knöchel, Thorsten; Musil, Djordje; Leuthner, Birgitta; Zenke, Frank
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 3(2017)
Page Start:
551
Record Type:
Journal Article
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5. R399E, A Mutated Form of Growth and Differentiation Factor 5, for Disease Modification of Osteoarthritis. Issue 3 (15th December 2022)

Authors:
Gigout, Anne; Werkmann, Daniela; Menges, Stephanie; Brenneis, Christian; Henson, Frances; Cowan, Kyra J.; Musil, Djordje; Thudium, Christian S.; Gühring, Hans; Michaelis, Martin; Kleinschmidt‐Doerr, Kerstin
Journal:
Arthritis & rheumatology
Issue:
Volume 75:Issue 3(2023)
Page Start:
375
Record Type:
Journal Article
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6. Structure-kinetic relationship reveals the mechanism of selectivity of FAK inhibitors over PYK2. Issue 5 (20th May 2021)

Authors:
Berger, Benedict-Tilman; Amaral, Marta; Kokh, Daria B.; Nunes-Alves, Ariane; Musil, Djordje; Heinrich, Timo; Schröder, Martin; Neil, Rebecca; Wang, Jing; Navratilova, Iva; Bomke, Joerg; Elkins, Jonathan M.; Müller, Susanne; Frech, Matthias; Wade, Rebecca C.; Knapp, Stefan
Journal:
Cell chemical biology
Issue:
Volume 28:Issue 5(2021)
Page Start:
686
Record Type:
Journal Article
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7. Zeitaufgelöst und markerfrei gemessene ligandeninduzierte Konformationsänderungen von HSP90 – hin zu einem Konformationsaktivitätsscreening für die Wirkstoffentwicklung. (3rd July 2018)

Authors:
Güldenhaupt, Jörn; Amaral, Marta; Kötting, Carsten; Schartner, Jonas; Musil, Djordje; Frech, Matthias; Gerwert, Klaus
Journal:
Angewandte Chemie
Issue:
Volume 130:Number 31(2018)
Page Start:
10103
Record Type:
Journal Article
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