1. Discovery and optimization of novel constrained pyrrolopyridone BET family inhibitors. Issue 10 (1st June 2018) Authors: Fidanze, Steven D.; Liu, Dachun; Mantei, Robert A.; Hasvold, Lisa A.; Pratt, John K.; Sheppard, George S.; Wang, Le; Holms, James H.; Dai, Yujia; Aguirre, Ana; Bogdan, Andrew; Dietrich, Justin D.; Marjanovic, Jasmina; Park, Chang H.; Hutchins, Charles W.; Lin, Xiaoyu; Bui, Mai H.; Huang, Xiaoli; ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 10(2018) Page Start: 1804 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Methylpyrrole inhibitors of BET bromodomains. Issue 10 (15th May 2017) Authors: Hasvold, Lisa A.; Sheppard, George S.; Wang, Le; Fidanze, Steven D.; Liu, Dachun; Pratt, John K.; Mantei, Robert A.; Wada, Carol K.; Hubbard, Robbert; Shen, Yu; Lin, Xiaoyu; Huang, Xiaoli; Warder, Scott E.; Wilcox, Denise; Li, Leiming; Buchanan, F. Greg; Smithee, Lauren; Albert, Daniel H.; Magoc,... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 10(2017) Page Start: 2225 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗