1. A small molecule inhibitor of HER3: a proof-of-concept study. Issue 17 (10th September 2020) Authors: Colomba, Audrey; Fitzek, Martina; George, Roger; Weitsman, Gregory; Roberts, Selene; Zanetti-Domingues, Laura; Hirsch, Michael; Rolfe, Daniel J.; Mehmood, Shahid; Madin, Andrew; Claus, Jeroen; Kjaer, Svend; Snijders, Ambrosius P.; Ng, Tony; Martin-Fernandez, Marisa; Smith, David M.; Parker, Peter J. Journal: Biochemical journal Issue: Volume 477:Issue 17(2020) Page Start: 3329 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Demonstration of the utility of DOS-derived fragment libraries for rapid hit derivatisation in a multidirectional fashion. Issue 39 (21st May 2020) Authors: Kidd, Sarah L.; Fowler, Elaine; Reinhardt, Till; Compton, Thomas; Mateu, Natalia; Newman, Hector; Bellini, Dom; Talon, Romain; McLoughlin, Joseph; Krojer, Tobias; Aimon, Anthony; Bradley, Anthony; Fairhead, Michael; Brear, Paul; Díaz-Sáez, Laura; McAuley, Katherine; Sore, Hannah F.; Madin, Andrew... Journal: Chemical science Issue: Volume 11:Issue 39(2020) Page Start: 10792 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of a selective c-MET inhibitor with a novel binding mode. (1st November 2022) Authors: Collie, Gavin W.; Barlind, Louise; Bazzaz, Sana; Börjesson, Ulf; Dale, Ian L.; Disch, Jeremy S.; Habeshian, Sevan; Jetson, Rachael; Khurana, Puneet; Madin, Andrew; Michaelides, Iacovos N.; Peng, Ling; Snijder, Arjan; Stubbs, Christopher J. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 75(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Highly efficient on-DNA amide couplings promoted by micelle forming surfactants for the synthesis of DNA encoded libraries. Issue 27 (22nd June 2021) Authors: Hunter, James H.; Anderson, Matthew J.; Castan, Isaline F. S. F.; Graham, Jessica S.; Salvini, Catherine L. A.; Stanway-Gordon, Harriet A.; Crawford, James J.; Madin, Andrew; Pairaudeau, Garry; Waring, Michael J. Journal: Chemical science Issue: Volume 12:Issue 27(2021) Page Start: 9475 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Identification and optimisation of a series of tetrahydrobenzotriazoles as metabotropic glutamate receptor 5-selective positive allosteric modulators that improve performance in a preclinical model of cognition. Issue 24 (15th December 2015) Authors: Ellard, John M.; Madin, Andrew; Philps, Oliver; Hopkin, Mark; Henderson, Scott; Birch, Louise; O'Connor, Desmond; Arai, Tohru; Takase, Kazuma; Morgan, Louise; Reynolds, David; Talma, Sonia; Howley, Eimear; Powney, Ben; Payne, Andrew H.; Hall, Adrian; Gartlon, Jane E.; Dawson, Lee A.; Castro, Luis... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 24(2015) Page Start: 5792 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Partially Saturated Bicyclic Heteroaromatics as an sp3‐Enriched Fragment Collection. (6th September 2016) Authors: Twigg, David G.; Kondo, Noriyasu; Mitchell, Sophie L.; Galloway, Warren R. J. D.; Sore, Hannah F.; Madin, Andrew; Spring, David R. Journal: Angewandte Chemie Issue: Volume 128:Number 40(2016) Page Start: 12667 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Partially Saturated Bicyclic Heteroaromatics as an sp3‐Enriched Fragment Collection. Issue 40 (6th September 2016) Authors: Twigg, David G.; Kondo, Noriyasu; Mitchell, Sophie L.; Galloway, Warren R. J. D.; Sore, Hannah F.; Madin, Andrew; Spring, David R. Journal: Angewandte Chemie international edition Issue: Volume 55:Issue 40(2016) Page Start: 12479 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Scope of on-DNA nucleophilic aromatic substitution on weakly-activated heterocyclic substrates for the synthesis of DNA-encoded libraries. (1st June 2022) Authors: Castan, Isaline F.S.F.; Madin, Andrew; Pairaudeau, Garry; Waring, Michael J. Journal: Bioorganic & medicinal chemistry Issue: Volume 63(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Synthesis of Structurally Diverse N‐Substituted Quaternary‐Carbon‐Containing Small Molecules from α, α‐Disubstituted Propargyl Amino Esters. Issue 51 (13th August 2018) Authors: Mateu, Natalia; Kidd, Sarah L.; Kalash, Leen; Sore, Hannah F.; Madin, Andrew; Bender, Andreas; Spring, David R. Journal: Chemistry Issue: Volume 24:Issue 51(2018) Page Start: 13681 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Tool inhibitors and assays to interrogate the biology of the TRAF2 and NCK interacting kinase. Issue 15 (1st August 2019) Authors: Read, Jon; Collie, Iain T.; Nguyen-McCarty, Michelle; Lucaj, Christopher; Robinson, James; Conway, Leslie; Mukherjee, Jayanta; McCall, Eileen; Donohoe, Gerard; Flavell, Elizabeth; Peciak, Karolina; Warwicker, Juli; Dix, Carly; Van den Hoven, Bernard G.; Madin, Andrew; Brown, Dean G.; Moss, Stephe... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 29:Issue 15(2019) Page Start: 1962 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗