1. Discovery of DC_H31 as potential mutant IDH1 inhibitor through NADPH-based high throughput screening. Issue 15 (1st August 2019) Authors: Duan, Zhe; Liu, Jingqiu; Niu, Liping; Wang, Jun; Feng, Mingqian; Chen, Hua; Luo, Cheng Journal: Bioorganic & medicinal chemistry Issue: Volume 27:Issue 15(2019) Page Start: 3229 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of potent DOT1L inhibitors by AlphaLISA based High Throughput Screening assay. Issue 8 (1st May 2018) Authors: Song, Yakai; Li, Linjuan; Chen, Yantao; Liu, Jingqiu; Xiao, Senhao; Lian, Fulin; Zhang, Naixia; Ding, Hong; Zhang, Yuanyuan; Chen, Kaixian; Jiang, Hualiang; Zhang, Chenhua; Liu, Yu-Chih; Chen, Shijie; Luo, Cheng Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 8(2018) Page Start: 1751 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Identification of a novel selective small-molecule inhibitor of protein arginine methyltransferase 5 (PRMT5) by virtual screening, resynthesis and biological evaluations. Issue 9 (15th May 2018) Authors: Zhu, Kongkai; Jiang, Chengshi; Tao, Hongrui; Liu, Jingqiu; Zhang, Hua; Luo, Cheng Journal: Bioorganic & medicinal chemistry letters Issue: Volume 28:Issue 9(2018) Page Start: 1476 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Identification of novel EZH2 inhibitors through pharmacophore-based virtual screening and biological assays. Issue 15 (1st August 2016) Authors: Wu, Yunlong; Hu, Junchi; Ding, Hong; Chen, Limin; Zhang, Yuanyuan; Liu, Rongfeng; Xu, Pan; Du, Daohai; Lu, Wenchao; Liu, Jingqiu; Liu, Yan; Liu, Yu-Chih; Lu, Junyan; Zhang, Jin; Yao, Zhiyi; Luo, Cheng Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 15(2016) Page Start: 3813 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Integrin β3 Deficiency Results in Hypertriglyceridemia via Disrupting LPL (Lipoprotein Lipase) Secretion. Issue 5 (May 2020) Authors: Xiao, Bing; Mao, Jianhua; Sun, Boyang; Zhang, Wei; Wang, Yun; Wang, Pengran; Ruan, Zheng; Xi, Wenda; Li, Huiyuan; Zhou, Jingyi; Lu, Yide; Ding, Qiulan; Wang, Xuefeng; Liu, Jingqiu; Yan, Jinsong; Luo, Cheng; Shi, Xiaofeng; Yang, Renchi; Xi, Xiaodong Journal: Arteriosclerosis, thrombosis, and vascular biology Issue: Volume 40:Issue 5(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Licochalcone A suppresses the proliferation of sarcoma HT-1080 cells, as a selective R132C mutant IDH1 inhibitor. Issue 2 (15th January 2020) Authors: Hu, Chujiao; Zuo, Yu; Liu, Jingqiu; Xu, Heng; Liao, Weike; Dang, Yongjun; Luo, Cheng; Tang, Lei; Zhang, Hao Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 2(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Targeting the RT loop of Src SH3 in Platelets Prevents Thrombosis without Compromising Hemostasis. Issue 7 (12th January 2022) Authors: Mao, Jianhua; Zhu, Kongkai; Long, Zhangbiao; Zhang, Huimin; Xiao, Bing; Xi, Wenda; Wang, Yun; Huang, Jiansong; Liu, Jingqiu; Shi, Xiaofeng; Jiang, Hao; Lu, Tian; Wen, Yi; Zhang, Naixia; Meng, Qian; Zhou, Hu; Ruan, Zheng; Wang, Jin; Luo, Cheng; Xi, Xiaodong Journal: Advanced science Issue: Volume 9:Issue 7(2022) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. The discovery of a non-competitive GOT1 inhibitor, hydralazine hydrochloride, via a coupling reaction-based high-throughput screening assay. (1st October 2022) Authors: Wu, Qiqi; Sun, Zhongya; Chen, Zhifeng; Liu, Jingqiu; Ding, Hong; Luo, Cheng; Wang, Mingliang; Du, Daohai Journal: Bioorganic & medicinal chemistry letters Issue: Volume 73(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗