1. Discovery and structure-based design of 4, 6-diaminonicotinamides as potent and selective IRAK4 inhibitors. Issue 21 (1st November 2017) Authors: Bhide, Rajeev S.; Keon, Alec; Weigelt, Carolyn; Sack, John S.; Schmidt, Robert J.; Lin, Shuqun; Xiao, Hai-Yun; Spergel, Steven H.; Kempson, James; Pitts, William J.; Carman, Julie; Poss, Michael A. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 21(2017) Page Start: 4908 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of highly potent, selective, covalent inhibitors of JAK3. Issue 20 (15th October 2017) Authors: Kempson, James; Ovalle, Damaso; Guo, Junqing; Wrobleski, Stephen T.; Lin, Shuqun; Spergel, Steven H.; Duan, James J.-W.; Jiang, Bin; Lu, Zhonghui; Das, Jagabandhu; Yang, Bingwei V.; Hynes, John; Wu, Hong; Tokarski, John; Sack, John S.; Khan, Javed; Schieven, Gary; Blatt, Yuval; Chaudhry, Charu; S... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 20(2017) Page Start: 4622 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗