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Author/Creator Leftheris, Katerina

1. Brain penetrant liver X receptor (LXR) modulators based on a 2, 4, 5, 6-tetrahydropyrrolo[3, 4-c]pyrazole core. Issue 20 (15th October 2016)

Authors:
Tice, Colin M.; Noto, Paul B.; Fan, Kristi Yi; Zhao, Wei; Lotesta, Stephen D.; Dong, Chengguo; Marcus, Andrew P.; Zheng, Ya-Jun; Chen, Guozhou; Wu, Zhongren; Van Orden, Rebecca; Zhou, Jing; Bukhtiyarov, Yuri; Zhao, Yi; Lipinski, Kerri; Howard, Lamont; Guo, Joan; Kandpal, Geeta; Meng, Shi; Hardy, ...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 20(2016)
Page Start:
5044
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

2. Brain penetrant liver X receptor (LXR) modulators based on a 2, 4, 5, 6-tetrahydropyrrolo[3, 4-c]pyrazole core. Issue 20 (15th October 2016)

Authors:
Tice, Colin M.; Noto, Paul B.; Fan, Kristi Yi; Zhao, Wei; Lotesta, Stephen D.; Dong, Chengguo; Marcus, Andrew P.; Zheng, Ya-Jun; Chen, Guozhou; Wu, Zhongren; Van Orden, Rebecca; Zhou, Jing; Bukhtiyarov, Yuri; Zhao, Yi; Lipinski, Kerri; Howard, Lamont; Guo, Joan; Kandpal, Geeta; Meng, Shi; Hardy, ...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 20(2016)
Page Start:
5044
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

3. Discovery of BI 135585, an in vivo efficacious oxazinanone-based 11β hydroxysteroid dehydrogenase type 1 inhibitor. Issue 14 (15th July 2017)

Authors:
Zhuang, Linghang; Tice, Colin M.; Xu, Zhenrong; Zhao, Wei; Cacatian, Salvacion; Ye, Yuan-Jie; Singh, Suresh B.; Lindblom, Peter; McKeever, Brian M.; Krosky, Paula M.; Zhao, Yi; Lala, Deepak; Kruk, Barbara A.; Meng, Shi; Howard, Lamont; Johnson, Judith A.; Bukhtiyarov, Yuri; Panemangalore, Reshma;...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 25:Issue 14(2017)
Page Start:
3649
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗

4. Identification of spirooxindole and dibenzoxazepine motifs as potent mineralocorticoid receptor antagonists. Issue 6 (15th March 2016)

Authors:
Lotesta, Stephen D.; Marcus, Andrew P.; Zheng, Yajun; Leftheris, Katerina; Noto, Paul B.; Meng, Shi; Kandpal, Geeta; Chen, Guozhou; Zhou, Jing; McKeever, Brian; Bukhtiyarov, Yuri; Zhao, Yi; Lala, Deepak S.; Singh, Suresh B.; McGeehan, Gerard M.
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 24:Issue 6(2016)
Page Start:
1384
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗