1. Discovery of novel 7-azaindoles as PDK1 inhibitors. Issue 13 (1st July 2016) Authors: Wucherer-Plietker, Margarita; Merkul, Eugen; Müller, Thomas J.J.; Esdar, Christina; Knöchel, Thorsten; Heinrich, Timo; Buchstaller, Hans-Peter; Greiner, Hartmut; Dorsch, Dieter; Finsinger, Dirk; Calderini, Michel; Bruge, David; Grädler, Ulrich Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 13(2016) Page Start: 3073 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Novel reversible methionine aminopeptidase-2 (MetAP-2) inhibitors based on purine and related bicyclic templates. Issue 3 (1st February 2017) Authors: Heinrich, Timo; Buchstaller, Hans-Peter; Cezanne, Bertram; Rohdich, Felix; Bomke, Jörg; Friese-Hamim, Manja; Krier, Mireille; Knöchel, Thorsten; Musil, Djordje; Leuthner, Birgitta; Zenke, Frank Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 3(2017) Page Start: 551 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗