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Author/Creator Kawatkar, Sameer

1. EED-Targeted PROTACs Degrade EED, EZH2, and SUZ12 in the PRC2 Complex. Issue 1 (16th January 2020)

Authors:
Hsu, Jessie Hao-Ru; Rasmusson, Timothy; Robinson, James; Pachl, Fiona; Read, Jon; Kawatkar, Sameer; O' Donovan, Daniel H.; Bagal, Sharan; Code, Erin; Rawlins, Philip; Argyrou, Argyrides; Tomlinson, Ronald; Gao, Ning; Zhu, Xiahui; Chiarparin, Elisabetta; Jacques, Kelly; Shen, Minhui; Woods, Haley;...
Journal:
Cell chemical biology
Issue:
Volume 27:Issue 1(2020)
Page Start:
41
Record Type:
Journal Article
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2. Free energy perturbation in the design of EED ligands as inhibitors of polycomb repressive complex 2 (PRC2) methyltransferase. (1st May 2021)

Authors:
O' Donovan, Daniel H.; Gregson, Clare; Packer, Martin J.; Greenwood, Ryan; Pike, Kurt G.; Kawatkar, Sameer; Bloecher, Andrew; Robinson, James; Read, Jon; Code, Erin; Hsu, Jessie Hao-Ru; Shen, Minhui; Woods, Haley; Barton, Peter; Fillery, Shaun; Williamson, Beth; Rawlins, Philip B.; Bagal, Sharan K.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 39(2021)
Page Start:
Record Type:
Journal Article
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3. Identification of azabenzimidazoles as potent JAK1 selective inhibitors. Issue 1 (1st January 2016)

Authors:
Vasbinder, Melissa M.; Alimzhanov, Marat; Augustin, Martin; Bebernitz, Geraldine; Bell, Kirsten; Chuaqui, Claudio; Deegan, Tracy; Ferguson, Andrew D.; Goodwin, Kelly; Huszar, Dennis; Kawatkar, Aarti; Kawatkar, Sameer; Read, Jon; Shi, Jie; Steinbacher, Stefan; Steuber, Holger; Su, Qibin; Toader, D...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 1(2016)
Page Start:
60
Record Type:
Journal Article
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4. Novel potent and selective pyrazolylpyrimidine-based SYK inhibitors. Issue 22 (15th November 2020)

Authors:
Barlaam, Bernard; Boiko, Scott; Boyd, Scott; Dry, Hannah; Gingipalli, Lakshmaiah; Ikeda, Timothy; Johnson, Tony; Kawatkar, Sameer; Lorthioir, Olivier; Pike, Andy; Pollard, Hannah; Read, Jon; Su, Qibin; Wang, Haiyun; Wang, Huimin; Wang, Lianghe; Wang, Peng; Edmondson, Scott D.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 22(2020)
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Record Type:
Journal Article
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5. Optimization of a series of potent, selective and orally bioavailable SYK inhibitors. Issue 19 (1st October 2020)

Authors:
Grimster, Neil P.; Gingipalli, Lakshmaiah; Barlaam, Bernard; Su, Qibin; Zheng, XiaoLan; Watson, David; Wang, Haixia; Simpson, Iain; Pike, Andy; Balazs, Amber; Boiko, Scott; Ikeda, Timothy P.; Impastato, Anna C.; Jones, Natalie H.; Kawatkar, Sameer; Kemmitt, Paul; Lamont, Scott; Patel, Joe; Read, ...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 19(2020)
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Record Type:
Journal Article
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