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Author/Creator Jespers, Willem

1. A2B adenosine receptor antagonists rescue lymphocyte activity in adenosine-producing patient-derived cancer models. Issue 5 (17th May 2022)

Authors:
Tay, Apple Hui Min; Prieto-Díaz, Rubén; Neo, Shiyong; Tong, Le; Chen, Xinsong; Carannante, Valentina; Önfelt, Björn; Hartman, Johan; Haglund, Felix; Majellaro, Maria; Azuaje, Jhonny; Garcia-Mera, Xerardo; Brea, Jose M; Loza, Maria I; Jespers, Willem; Gutierrez-de-Teran, Hugo; Sotelo, Eddy; Lundqv...
Journal:
Journal for immunotherapy of cancer
Issue:
Volume 10:Issue 5(2022)
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Record Type:
Journal Article
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2. Cancer‐related somatic mutations alter adenosine A1 receptor pharmacology—A focus on mutations in the loops and C‐terminus. Issue 6 (23rd May 2022)

Authors:
Wang, Xuesong; Jespers, Willem; de Waal, Just J.; Wolff, Kim A. N.; van Uden, Liedeke; IJzerman, Adriaan P.; van Westen, Gerard J. P.; Heitman, Laura H.
Journal:
FASEB journal
Issue:
Volume 36:Issue 6(2022)
Page Start:
n/a
Record Type:
Journal Article
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3. Development of subtype-selective covalent ligands for the adenosine A2B receptor by tuning the reactive group. Issue 7 (30th June 2022)

Authors:
Beerkens, Bert L. H.; Wang, Xuesong; Avgeropoulou, Maria; Adistia, Lisa N.; van Veldhoven, Jacobus P. D.; Jespers, Willem; Liu, Rongfang; Heitman, Laura H.; IJzerman, Adriaan P.; van der Es, Daan
Journal:
RSC medicinal chemistry
Issue:
Volume 13:Issue 7(2022)
Page Start:
850
Record Type:
Journal Article
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4. Structural Mapping of Adenosine Receptor Mutations: Ligand Binding and Signaling Mechanisms. (January 2018)

Authors:
Jespers, Willem; Schiedel, Anke C.; Heitman, Laura H.; Cooke, Robert M.; Kleene, Lisa; van Westen, Gerard J.P.; Gloriam, David E.; Müller, Christa E.; Sotelo, Eddy; Gutiérrez-de-Terán, Hugo
Journal:
Trends in pharmacological sciences
Issue:
Volume 39:Number 1(2018)
Page Start:
75
Record Type:
Journal Article
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5. X‐Ray Crystallography and Free Energy Calculations Reveal the Binding Mechanism of A2A Adenosine Receptor Antagonists. (22nd July 2020)

Authors:
Jespers, Willem; Verdon, Grégory; Azuaje, Jhonny; Majellaro, Maria; Keränen, Henrik; García‐Mera, Xerardo; Congreve, Miles; Deflorian, Francesca; de Graaf, Chris; Zhukov, Andrei; Doré, Andrew S.; Mason, Jonathan S.; Åqvist, Johan; Cooke, Robert M.; Sotelo, Eddy; Gutiérrez‐de‐Terán, Hugo
Journal:
Angewandte Chemie
Issue:
Volume 132:Number 38(2020)
Page Start:
16679
Record Type:
Journal Article
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6. X‐Ray Crystallography and Free Energy Calculations Reveal the Binding Mechanism of A2A Adenosine Receptor Antagonists. Issue 38 (22nd July 2020)

Authors:
Jespers, Willem; Verdon, Grégory; Azuaje, Jhonny; Majellaro, Maria; Keränen, Henrik; García‐Mera, Xerardo; Congreve, Miles; Deflorian, Francesca; de Graaf, Chris; Zhukov, Andrei; Doré, Andrew S.; Mason, Jonathan S.; Åqvist, Johan; Cooke, Robert M.; Sotelo, Eddy; Gutiérrez‐de‐Terán, Hugo
Journal:
Angewandte Chemie international edition
Issue:
Volume 59:Issue 38(2020)
Page Start:
16536
Record Type:
Journal Article
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