1. Design and synthesis of new homo and hetero bis-piperazinyl-1-propanone derivatives as 5-HT7R selective ligands over 5-HT1AR. Issue 16 (15th August 2016) Authors: Intagliata, Sebastiano; Modica, Maria N.; Pittalà, Valeria; Salerno, Loredana; Siracusa, Maria A.; Cagnotto, Alfredo; Salmona, Mario; Romeo, Giuseppe Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 16(2016) Page Start: 4052 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of 3‐(2‐aminoethyl)‐thiazolidine‐2, 4‐diones as a novel chemotype of sigma‐1 receptor ligands. (25th April 2022) Authors: Elkholy, Nada; Abdelwaly, Ahmad; Mohamed, Karim; Amata, Emanuele; Lombino, Jessica; Cosentino, Giuseppe; Intagliata, Sebastiano; Helal, Mohamed A. Journal: Chemical biology & drug design Issue: Volume 100:Number 1(2022) Page Start: 25 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of SI 1/20 and SI 1/22 as Mutual Prodrugs of 5‐Fluorouracil and Imidazole‐Based Heme Oxygenase 1 Inhibitor with Improved Cytotoxicity in DU145 Prostate Cancer Cells. (24th February 2023) Authors: Salerno, Loredana; Sorrenti, Valeria; Pittalà, Valeria; Consoli, Valeria; Modica, Maria N.; Romeo, Giuseppe; Marrazzo, Agostino; Giuliano, Michela; Zajdel, Paweł; Vanella, Luca; Intagliata, Sebastiano Journal: ChemMedChem Issue: Volume 18:Number 8(2023) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. In vitro and in silico analysis of imatinib analogues as anti-Trypanosoma cruzi drug candidates. Issue 4 (12th April 2023) Authors: Nesic de Freitas, Luca S. F.; da Silva, Cristiane França; Intagliata, Sebastiano; Amata, Emanuele; Salerno, Loredana; Soeiro, Maria de Nazaré Correia Journal: Parasitology Issue: Volume 150:Issue 4(2023) Page Start: 359 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Mutual Prodrugs of 5‐Fluorouracil: From a Classic Chemotherapeutic Agent to Novel Potential Anticancer Drugs. (7th September 2021) Authors: Ciaffaglione, Valeria; Modica, Maria N.; Pittalà, Valeria; Romeo, Giuseppe; Salerno, Loredana; Intagliata, Sebastiano Journal: ChemMedChem Issue: Volume 16:Number 23(2021) Page Start: 3496 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. New N- and O-arylpiperazinylalkyl pyrimidines and 2-methylquinazolines derivatives as 5-HT7 and 5-HT1A receptor ligands: Synthesis, structure-activity relationships, and molecular modeling studies. Issue 3 (1st February 2017) Authors: Intagliata, Sebastiano; Modica, Maria N.; Pittalà, Valeria; Salerno, Loredana; Siracusa, Maria A.; Cagnotto, Alfredo; Salmona, Mario; Kurczab, Rafał; Romeo, Giuseppe Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 3(2017) Page Start: 1250 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Novel mutual prodrug of 5-fluorouracil and heme oxygenase-1 inhibitor (5-FU/HO-1 hybrid): design and preliminary in vitro evaluation. (1st January 2021) Authors: Salerno, Loredana; Vanella, Luca; Sorrenti, Valeria; Consoli, Valeria; Ciaffaglione, Valeria; Fallica, Antonino N.; Canale, Vittorio; Zajdel, Paweł; Pignatello, Rosario; Intagliata, Sebastiano Journal: Journal of enzyme inhibition and medicinal chemistry Issue: Volume 36:Number 1(2021) Page Start: 1377 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Structure-activity relationships of mixed σ1R/σ2R ligands with antiproliferative and anticancer effects. (1st November 2022) Authors: Fallica, Antonino N.; Ciaffaglione, Valeria; Modica, Maria N.; Pittalà, Valeria; Salerno, Loredana; Amata, Emanuele; Marrazzo, Agostino; Romeo, Giuseppe; Intagliata, Sebastiano Journal: Bioorganic & medicinal chemistry Issue: Volume 73(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Synthesis and binding properties of new long-chain 4-substituted piperazine derivatives as 5-HT1A and 5-HT7 receptor ligands. Issue 7 (1st April 2015) Authors: Modica, Maria N.; Intagliata, Sebastiano; Pittalà, Valeria; Salerno, Loredana; Siracusa, Maria A.; Cagnotto, Alfredo; Salmona, Mario; Romeo, Giuseppe Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 7(2015) Page Start: 1427 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗