1. Discovery of novel 2′, 4′-dimethyl-[4, 5′-bithiazol]-2-yl amino derivatives as orally bioavailable TRPV4 antagonists for the treatment of pain: Part 1. Issue 20 (15th October 2016) Authors: Tsuno, Naoki; Yukimasa, Akira; Yoshida, Osamu; Ichihashi, Yusuke; Inoue, Takatsugu; Ueno, Tatsuhiko; Yamaguchi, Hiroki; Matsuda, Hidetoshi; Funaki, Satoko; Yamanada, Natsue; Tanimura, Miki; Nagamatsu, Daiki; Nishimura, Yoko; Ito, Tetsuji; Soga, Masahiko; Horita, Narumi; Yamamoto, Miyuki; Hinata, ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 20(2016) Page Start: 4930 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of novel 2′, 4′-dimethyl-[4, 5′-bithiazol]-2-yl amino derivatives as orally bioavailable TRPV4 antagonists for the treatment of pain: Part 2. Issue 20 (15th October 2016) Authors: Tsuno, Naoki; Yukimasa, Akira; Yoshida, Osamu; Suzuki, Shinji; Nakai, Hiromi; Ogawa, Tomoyuki; Fujiu, Motohiro; Takaya, Kenji; Nozu, Azusa; Yamaguchi, Hiroki; Matsuda, Hidetoshi; Funaki, Satoko; Nishimura, Yoko; Ito, Tetsuji; Nagamatsu, Daiki; Asaki, Toshiyuki; Horita, Narumi; Yamamoto, Miyuki; H... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 20(2016) Page Start: 4936 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Pharmacological evaluation of novel (6-aminopyridin-3-yl)(4-(pyridin-2-yl)piperazin-1-yl) methanone derivatives as TRPV4 antagonists for the treatment of pain. Issue 7 (1st April 2017) Authors: Tsuno, Naoki; Yukimasa, Akira; Yoshida, Osamu; Suzuki, Shinji; Nakai, Hiromi; Ogawa, Tomoyuki; Fujiu, Motohiro; Takaya, Kenji; Nozu, Azusa; Yamaguchi, Hiroki; Matsuda, Hidetoshi; Funaki, Satoko; Yamanada, Natsue; Tanimura, Miki; Nagamatsu, Daiki; Asaki, Toshiyuki; Horita, Narumi; Yamamoto, Miyuki... Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 7(2017) Page Start: 2177 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Sensitization of transient receptor potential vanilloid 4 and increasing its endogenous ligand 5, 6-epoxyeicosatrienoic acid in rats with monoiodoacetate-induced osteoarthritis. Issue 5 (May 2018) Authors: Hinata, Mikie; Imai, Sunao; Sanaki, Takao; Tsuchida, Junji; Yoshioka, Takeshi; Higashino, Kenichi; Yamamoto, Miyuki; Imai, Masayuki; Soga, Masahiko; Horita, Narumi; Fukuda, Isao; Ikeda, Minoru; Yamane, Shoji; Morita, Atsushi; Kanemasa, Toshiyuki; Sakaguchi, Gaku; Hasegawa, Minoru; Minami, Masabum... Journal: Pain Issue: Volume 159:Issue 5(2018) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗