1. Design, synthesis and evaluation of a novel series of inhibitors reversing P‐glycoprotein‐mediated multidrug resistance. (14th June 2018) Authors: Ghaleb, Hesham; Li, Huilan; Kairuki, Mutta; Qiu, Qianqian; Bi, Xinzhou; Liu, Chunxia; Liao, Chen; Li, Jieming; Hezam, Kamal; Huang, Wenlong; Qian, Hai Journal: Chemical biology & drug design Issue: Volume 92:Number 3(2018) Page Start: 1708 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Designed P-glycoprotein inhibitors with triazol-tetrahydroisoquinoline-core increase doxorubicin-induced mortality in multidrug resistant K562/A02 cells. Issue 15 (1st August 2019) Authors: Kairuki, Mutta; Qiu, Qianqian; Pan, Miaobo; Li, Qifei; Zhou, Jiaqi; Ghaleb, Hesham; Huang, Wenlong; Qian, Hai; Jiang, Cheng Journal: Bioorganic & medicinal chemistry Issue: Volume 27:Issue 15(2019) Page Start: 3347 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Phenylquinoline transient receptor potential vanilloid 1 antagonists for the treatment of pain: Discovery of 1-(2-phenylquinoline-4-carbonyl)-N-(4-(trifluoromethyl)phenyl)pyrrolidine-3-carboxamide. Issue 4 (15th February 2018) Authors: Liao, Chen; Liu, Yan; Liu, Chunxia; Zhou, Jiaqi; Li, Huilan; Wang, Nasi; Li, Jieming; Liu, Taiyu; Ghaleb, Hesham; Huang, Wenlong; Qian, Hai Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 4(2018) Page Start: 845 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗