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Author/Creator Gehling, Victor S.

1. Corrigendum to "Development of methyl isoxazoleazepines as inhibitors of BET" [Bioorg. Med. Chem. Lett. 25/9 (2015) 1842–1848]. Issue 17 (1st September 2015)

Authors:
Hewitt, Michael C.; Leblanc, Yves; Gehling, Victor S.; Vaswani, Rishi G.; Côté, Alexandre; Nasveschuk, Christopher G.; Taylor, Alexander M.; Harmange, Jean-Christophe; Audia, James E.; Pardo, Eneida; Cummings, Rich; Joshi, Shivangi; Sandy, Peter; Mertz, Jennifer A.; Sims, Robert J.; Bergeron, Lou...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 17(2015)
Page Start:
3755
Record Type:
Journal Article
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2. Development of methyl isoxazoleazepines as inhibitors of BET. Issue 9 (1st May 2015)

Authors:
Hewitt, Michael C.; Leblanc, Yves; Gehling, Victor S.; Vaswani, Rishi G.; Côté, Alexandre; Nasveschuk, Christopher G.; Taylor, Alexander M.; Harmange, Jean-Christophe; Audia, James E.; Pardo, Eneida; Cummings, Rich; Joshi, Shivangi; Sandy, Peter; Mertz, Jennifer A.; Sims, Robert J.; Bergeron, Lou...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 9(2015)
Page Start:
1842
Record Type:
Journal Article
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3. Development of methyl isoxazoleazepines as inhibitors of BET. Issue 9 (1st May 2015)

Authors:
Hewitt, Michael C.; Leblanc, Yves; Gehling, Victor S.; Vaswani, Rishi G.; Côté, Alexandre; Nasveschuk, Christopher G.; Taylor, Alexander M.; Harmange, Jean-Christophe; Audia, James E.; Pardo, Eneida; Cummings, Rich; Joshi, Shivangi; Sandy, Peter; Mertz, Jennifer A.; Sims, Robert J.; Bergeron, Lou...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 9(2015)
Page Start:
1842
Record Type:
Journal Article
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Available online (eLD content is only available in our Reading Rooms) ↗

4. Discovery, design, and synthesis of indole-based EZH2 inhibitors. Issue 17 (1st September 2015)

Authors:
Gehling, Victor S.; Vaswani, Rishi G.; Nasveschuk, Christopher G.; Duplessis, Martin; Iyer, Priyadarshini; Balasubramanian, Srividya; Zhao, Feng; Good, Andrew C.; Campbell, Robert; Lee, Christina; Dakin, Les A.; Cook, Andrew S.; Gagnon, Alexandre; Harmange, Jean-Christophe; Audia, James E.; Cummi...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 17(2015)
Page Start:
3644
Record Type:
Journal Article
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5. From a novel HTS hit to potent, selective, and orally bioavailable KDM5 inhibitors. Issue 13 (1st July 2017)

Authors:
Liang, Jun; Labadie, Sharada; Zhang, Birong; Ortwine, Daniel F.; Patel, Snahel; Vinogradova, Maia; Kiefer, James R.; Mauer, Till; Gehling, Victor S.; Harmange, Jean-Christophe; Cummings, Richard; Lai, Tommy; Liao, Jiangpeng; Zheng, Xiaoping; Liu, Yichin; Gustafson, Amy; Van der Porten, Erica; Mao...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 27:Issue 13(2017)
Page Start:
2974
Record Type:
Journal Article
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6. Identification of potent, selective KDM5 inhibitors. Issue 17 (1st September 2016)

Authors:
Gehling, Victor S.; Bellon, Steven F.; Harmange, Jean-Christophe; LeBlanc, Yves; Poy, Florence; Odate, Shobu; Buker, Shane; Lan, Fei; Arora, Shilpi; Williamson, Kaylyn E.; Sandy, Peter; Cummings, Richard T.; Bailey, Christopher M.; Bergeron, Louise; Mao, Weifeng; Gustafson, Amy; Liu, Yichin; Vand...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 17(2016)
Page Start:
4350
Record Type:
Journal Article
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7. Lead optimization of a pyrazolo[1, 5-a]pyrimidin-7(4H)-one scaffold to identify potent, selective and orally bioavailable KDM5 inhibitors suitable for in vivo biological studies. Issue 16 (15th August 2016)

Authors:
Liang, Jun; Zhang, Birong; Labadie, Sharada; Ortwine, Daniel F.; Vinogradova, Maia; Kiefer, James R.; Gehling, Victor S.; Harmange, Jean-Christophe; Cummings, Richard; Lai, Tommy; Liao, Jiangpeng; Zheng, Xiaoping; Liu, Yichin; Gustafson, Amy; Van der Porten, Erica; Mao, Weifeng; Liederer, Bianca ...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 16(2016)
Page Start:
4036
Record Type:
Journal Article
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