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Author/Creator Gege, Christian

1. Discovery and optimization of new oxadiazole substituted thiazole RORγt inverse agonists through a bioisosteric amide replacement approach. Issue 12 (15th June 2020)

Authors:
Steeneck, Christoph; Gege, Christian; Kinzel, Olaf; Albers, Michael; Kleymann, Gerald; Schlüter, Thomas; Schulz, Andreas; Xue, Xiaohua; Cummings, Maxwell D.; Fourie, Anne M.; Leonard, Kristi A.; Scott, Brian; Edwards, James P.; Hoffmann, Thomas; Goldberg, Steven D.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 12(2020)
Page Start:
Record Type:
Journal Article
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3. Identification and biological evaluation of thiazole-based inverse agonists of RORγt. Issue 9 (15th May 2018)

Authors:
Gege, Christian; Cummings, Maxwell D.; Albers, Michael; Kinzel, Olaf; Kleymann, Gerald; Schlüter, Thomas; Steeneck, Christoph; Nelen, Marina I.; Milligan, Cindy; Spurlino, John; Xue, Xiaohua; Leonard, Kristi; Edwards, James P.; Fourie, Anne; Goldberg, Steven D.; Hoffmann, Thomas
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 9(2018)
Page Start:
1446
Record Type:
Journal Article
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4. Novel substituted isoxazole FXR agonists with cyclopropyl, hydroxycyclobutyl and hydroxyazetidinyl linkers: Understanding and improving key determinants of pharmacological properties. Issue 15 (1st August 2016)

Authors:
Kinzel, Olaf; Steeneck, Christoph; Schlüter, Thomas; Schulz, Andreas; Gege, Christian; Hahn, Ulrike; Hambruch, Eva; Hornberger, Martin; Spalwisz, Adriana; Frick, Katharina; Perović-Ottstadt, Sanja; Deuschle, Ulrich; Burnet, Michael; Kremoser, Claus
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 15(2016)
Page Start:
3746
Record Type:
Journal Article
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5. Optimization and biological evaluation of thiazole-bis-amide inverse agonists of RORγt. Issue 12 (15th June 2020)

Authors:
Gege, Christian; Albers, Michael; Kinzel, Olaf; Kleymann, Gerald; Schlüter, Thomas; Steeneck, Christoph; Hoffmann, Thomas; Xue, Xiaohua; Cummings, Maxwell D.; Spurlino, John; Milligan, Cynthia; Fourie, Anne M.; Edwards, James P.; Leonard, Kristi; Coe, Kevin; Scott, Brian; Pippel, Dan; Goldberg, S...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 12(2020)
Page Start:
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗