1. [2.2.1]-Bicyclic sultams as potent androgen receptor antagonists. Issue 23 (1st December 2016) Authors: Shan, Weifang; Balog, Aaron; Nation, Andrew; Zhu, Xiao; Chen, Jing; Cvijic, Mary Ellen; Geng, Jieping; Rizzo, Cheryl A.; Spires, Thomas; Attar, Ricardo M.; Obermeier, Mary; Traeger, Sarah; Dai, Jun; Zhang, Yingru; Galella, Michael; Trainor, George; Vite, Gregory D.; Gavai, Ashvinikumar V. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 23(2016) Page Start: 5707 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. BMS-871: A novel orally active pan-Notch inhibitor as an anticancer agent. Issue 9 (1st May 2015) Authors: Shan, Weifang; Balog, Aaron; Quesnelle, Claude; Gill, Patrice; Han, Wen-Ching; Norris, Derek; Mandal, Sunilkumar; Thiruvenkadam, Raja; Gona, Kiran Babu; Thiyagarajan, Kamalraj; Kandula, Sathiah; McGlinchey, Kelly; Menard, Krista; Wen, Mei-Li; Rose, Anne; White, Ronald; Guarino, Victor; Shen, Ding... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 9(2015) Page Start: 1905 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. BMS-871: A novel orally active pan-Notch inhibitor as an anticancer agent. Issue 9 (1st May 2015) Authors: Shan, Weifang; Balog, Aaron; Quesnelle, Claude; Gill, Patrice; Han, Wen-Ching; Norris, Derek; Mandal, Sunilkumar; Thiruvenkadam, Raja; Gona, Kiran Babu; Thiyagarajan, Kamalraj; Kandula, Sathiah; McGlinchey, Kelly; Menard, Krista; Wen, Mei-Li; Rose, Anne; White, Ronald; Guarino, Victor; Shen, Ding... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 9(2015) Page Start: 1905 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Development of BET inhibitors as potential treatments for cancer: A new carboline chemotype. (1st November 2021) Authors: Hill, Matthew D.; Quesnelle, Claude; Tokarski, John; Fang, Haiquan; Fanslau, Carolynn; Haarhoff, Zuzana; Kramer, Melissa; Madari, Shilpa; Wiebesiek, Amy; Morrison, John; Simmermacher-Mayer, Jean; Sinz, Michael; Westhouse, Richard; Xie, Chunshan; Zhao, Jiuqiao; Huang, Lisa; Sheriff, Steven; Yan, C... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 51(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Development of BET inhibitors as potential treatments for cancer: A search for structural diversity. (15th July 2021) Authors: Hill, Matthew D.; Fang, Haiquan; Tokarski, John; Fanslau, Carolynn; Haarhoff, Zuzana; Huang, Christine; Kramer, Melissa; Menard, Krista; Monereau, Laura; Morrison, John; Ranasinghe, Asoka; Shields, Eric E.; Tye, Ching Kim; Westhouse, Richard; Everlof, Gerry; Sheriff, Steven; Yan, Chunhong; Marsil... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 44(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗