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Author/Creator Galella, Michael A.

1. Discovery and synthesis of cyclohexenyl derivatives as modulators of CC chemokine receptor 2 activity. Issue 2 (15th January 2016)

Authors:
Brown, Gregory D.; Shi, Qing; Delucca, George V.; Batt, Douglas G.; Galella, Michael A.; Cvijic, Mary-Ellen; Liu, Rui-Qin; Qiu, Feng; Zhao, Qihong; Barrish, Joel C.; Carter, Percy H.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 26:Issue 2(2016)
Page Start:
662
Record Type:
Journal Article
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2. Discovery of (3S, 4S)-3-methyl-3-(4-fluorophenyl)-4-(4-(1, 1, 1, 3, 3, 3-hexafluoro-2-hydroxyprop-2-yl)phenyl)pyrrolidines as novel RORγt inverse agonists. Issue 17 (1st September 2020)

Authors:
Jiang, Bin; Duan, James J.-W.; Stachura, Sylwia; Karmakar, Ananta; Hemagiri, Hemalatha; Raut, Dhanya Kumar; Gupta, Arun Kumar; Weigelt, Carolyn A.; Khan, Javed; Sack, John S.; Wu, Dauh-Rurng; Yarde, Melissa; Shen, Ding-Ren; Galella, Michael A.; Mathur, Arvind; Zhao, Qihong; Salter-Cid, Luisa M.; ...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 17(2020)
Page Start:
Record Type:
Journal Article
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3. Identification of 6-hydroxy-5-phenyl sulfonylpyrimidin-4(1H)-one APJ receptor agonists. (15th October 2021)

Authors:
Tora, George; Jiang, Ji; Bostwick, Jeffrey S.; Gargalovic, Peter S.; Onorato, Joelle M.; Luk, Chiuwa E.; Generaux, Claudia; Xu, Carrie; Galella, Michael A.; Wang, Tao; He, Yan; Wexler, Ruth R.; Finlay, Heather J.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 50(2021)
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Record Type:
Journal Article
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4. Identification of bicyclic hexafluoroisopropyl alcohol sulfonamides as retinoic acid receptor-related orphan receptor gamma (RORγ/RORc) inverse agonists. Employing structure-based drug design to improve pregnane X receptor (PXR) selectivity. Issue 2 (15th January 2018)

Authors:
Gong, Hua; Weinstein, David S.; Lu, Zhonghui; Duan, James J.-W.; Stachura, Sylwia; Haque, Lauren; Karmakar, Ananta; Hemagiri, Hemalatha; Raut, Dhanya Kumar; Gupta, Arun Kumar; Khan, Javed; Camac, Dan; Sack, John S.; Pudzianowski, Andrew; Wu, Dauh-Rurng; Yarde, Melissa; Shen, Ding-Ren; Borowski, V...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 2(2018)
Page Start:
85
Record Type:
Journal Article
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Available online (eLD content is only available in our Reading Rooms) ↗