1. Corrigendum to "Design of selective PI3Kδ inhibitors using an iterative scaffold-hopping workflow" [Bioorg. Med. Chem. Lett. 29 (2019) 2575–2580]. Issue 16 (15th August 2020) Authors: Fradera, Xavier; Methot, Joey L.; Achab, Abdelghani; Christopher, Matthew; Altman, Michael D.; Zhou, Hua; McGowan, Meredeth A.; Kattar, Sam D.; Wilson, Kevin; Garcia, Yudith; Augustin, Martin A.; Lesburg, Charles A.; Shah, Sanjiv; Goldenblatt, Peter; Katz, Jason D. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 16(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of IDO1 inhibitors containing a decahydroquinoline, decahydro-1, 6-naphthyridine, or octahydro-1H-pyrrolo[3, 2-c]pyridine scaffold. (1st October 2021) Authors: Yu, Wensheng; Deng, Yongqi; Sloman, David; Li, Derun; Liu, Kun; Fradera, Xavier; Lesburg, Charles A.; Martinot, Theo; Doty, Amy; Ferguson, Heidi; Richard Miller, J.; Knemeyer, Ian; Otte, Karin; Vincent, Stella; Sciammetta, Nunzio; Jonathan Bennett, David; Han, Yongxin Journal: Bioorganic & medicinal chemistry letters Issue: Volume 49(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. SAR towards indoline and 3-azaindoline classes of IDO1 inhibitors. (1st September 2021) Authors: Yu, Wensheng; Deng, Yongqi; Hopkins, Brett; Huang, Xianhai; Sloman, David; Zhang, Hongjun; Li, Derun; McGowan, Meredeth A.; White, Catherine; Pu, Qinglin; Liu, Kun; Fradera, Xavier; Lesburg, Charles A.; Martinot, Theo; Doty, Amy; Ferguson, Heidi; Nickbarg, Elliott B.; Cheng, Mangeng; Geda, Prasan... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 47(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery and optimization of heteroaryl piperazines as potent and selective PI3Kδ inhibitors. Issue 1 (1st January 2020) Authors: Zhou, Hua; McGowan, Meredeth A.; Lipford, Kathryn; Christopher, Matthew; Fradera, Xavier; Witter, David; Lesburg, Charles A.; Li, Chaomin; Methot, Joey L.; Lampe, John; Achab, Abdelghani; Shaffer, Lynsey; Goldenblatt, Peter; Shah, Sanjiv; Bass, Alan; Schroeder, Gottfried; Chen, Dapeng; Zeng, Haoy... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 1(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Design of selective PI3Kδ inhibitors using an iterative scaffold-hopping workflow. Issue 18 (15th September 2019) Authors: Fradera, Xavier; Methot, Joey L.; Achab, Abdelghani; Christopher, Matthew; Altman, Michael D.; Zhou, Hua; McGowan, Meredeth A.; Kattar, Sam D.; Wilson, Kevin; Garcia, Yudith; Augustin, Martin A.; Lesburg, Charles A.; Shah, Sanjiv; Goldenblatt, Peter; Katz, Jason D. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 29:Issue 18(2019) Page Start: 2575 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. NMR Data‐Driven Docking of HDM2‐Inhibitor Complexes. (21st February 2022) Authors: Fradera, Xavier; Reutershan, Michael H.; Machacek, Michelle R.; Trotter, B. Wesley; McCoy, Mark A. Journal: Chembiochem Issue: Volume 23:Number 6(2022) Page Start: n/a Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. Development of High-Throughput Assays for Evaluation of Hematopoietic Progenitor Kinase 1 Inhibitors. (January 2021) Authors: Lacey, Brian M.; Xu, Zangwei; Chai, Xiaomei; Laskey, Jason; Fradera, Xavier; Mittal, Payal; Mishra, Sasmita; Piesvaux, Jennifer; Saradjian, Peter; Shaffer, Lynsey; Vassileva, Galya; Gerdt, Catherine; Wang, Yun; Ferguson, Heidi; Smith, Dustin M.; Ballard, Jeanine; Wells, Steven; Jain, Rishabh; Mue... Journal: SLAS discovery Issue: Volume 26:Number 1(2021) Page Start: 88 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. Overview of Methods and Strategies for Conducting Virtual Small Molecule Screening. Issue 3 (14th September 2017) Authors: Fradera, Xavier; Babaoglu, Kerim Journal: Current protocols in chemical biology Issue: Volume 9:Issue 3(2017) Page Start: 196 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
9. Discovery of a new series of PI3K-δ inhibitors from Virtual Screening. (15th June 2021) Authors: Fradera, Xavier; Deng, Qiaolin; Achab, Abdelganhi; Garcia, Yudith; Kattar, Solomon D.; McGowan, Meredeth A.; Methot, Joey L.; Wilson, Kevin; Zhou, Hua; Shaffer, Lynsey; Goldenblatt, Peter; Tong, Vincent; Augustin, Martin A; Altman, Michael D.; Lesburg, Charles A.; Shah, Sanjiv; Katz, Jason D. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 42(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
10. Repurposing a Histamine Detection Platform for High-Throughput Screening of Histidine Decarboxylase. (October 2018) Authors: Juang, Yu-Chi; Fradera, Xavier; Han, Yongxin; Partridge, Anthony William Journal: SLAS discovery Issue: Volume 23:Number 9(2018) Page Start: 974 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗