1. A small molecule inhibitor of HER3: a proof-of-concept study. Issue 17 (10th September 2020) Authors: Colomba, Audrey; Fitzek, Martina; George, Roger; Weitsman, Gregory; Roberts, Selene; Zanetti-Domingues, Laura; Hirsch, Michael; Rolfe, Daniel J.; Mehmood, Shahid; Madin, Andrew; Claus, Jeroen; Kjaer, Svend; Snijders, Ambrosius P.; Ng, Tony; Martin-Fernandez, Marisa; Smith, David M.; Parker, Peter J. Journal: Biochemical journal Issue: Volume 477:Issue 17(2020) Page Start: 3329 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Design of selective PI3Kα inhibitors starting from a promiscuous pan kinase scaffold. Issue 13 (1st July 2015) Authors: Barlaam, Bernard; Cosulich, Sabina; Fitzek, Martina; Green, Stephen; Harris, Craig S.; Hudson, Kevin; Lambert-van der Brempt, Christine; Ouvry, Gilles; Page, Ken; Ruston, Linette; Ward, Lara; Delouvrié, Bénédicte Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 13(2015) Page Start: 2679 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of 1-(4-(5-(5-amino-6-(5-tert-butyl-1, 3, 4-oxadiazol-2-yl)pyrazin-2-yl)-1-ethyl-1, 2, 4-triazol-3-yl)piperidin-1-yl)-3-hydroxypropan-1-one (AZD8835): A potent and selective inhibitor of PI3Kα and PI3Kδ for the treatment of cancers. Issue 22 (15th November 2015) Authors: Barlaam, Bernard; Cosulich, Sabina; Delouvrié, Bénédicte; Ellston, Rebecca; Fitzek, Martina; Germain, Hervé; Green, Stephen; Hancox, Urs; Harris, Craig S.; Hudson, Kevin; Lambert-van der Brempt, Christine; Lebraud, Honorine; Magnien, Françoise; Lamorlette, Maryannick; Le Griffon, Antoine; Morgent... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 22(2015) Page Start: 5155 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery of a novel aminopyrazine series as selective PI3Kα inhibitors. Issue 13 (1st July 2017) Authors: Barlaam, Bernard; Cosulich, Sabina; Fitzek, Martina; Germain, Hervé; Green, Stephen; Hanson, Lyndsey L.; Harris, Craig S.; Hancox, Urs; Hudson, Kevin; Lambert-van der Brempt, Christine; Lamorlette, Maryannick; Magnien, Françoise; Ouvry, Gilles; Page, Ken; Ruston, Linette; Ward, Lara; Delouvrié, B... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 13(2017) Page Start: 3030 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Discovery of a series of 8-(1-phenylpyrrolidin-2-yl)-6-carboxamide-2-morpholino-4H-chromen-4-one as PI3Kβ/δ inhibitors for the treatment of PTEN-deficient tumours. Issue 9 (1st May 2017) Authors: Barlaam, Bernard; Cosulich, Sabina; Degorce, Sébastien; Ellston, Rebecca; Fitzek, Martina; Green, Stephen; Hancox, Urs; Lambert-van der Brempt, Christine; Lohmann, Jean-Jacques; Maudet, Mickaël; Morgentin, Rémy; Plé, Patrick; Ward, Lara; Warin, Nicolas Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 9(2017) Page Start: 1949 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Discovery of a series of 8-(2, 3-dihydro-1, 4-benzoxazin-4-ylmethyl)-2-morpholino-4-oxo-chromene-6-carboxamides as PI3Kβ/δ inhibitors for the treatment of PTEN-deficient tumours. Issue 9 (1st May 2016) Authors: Barlaam, Bernard; Cosulich, Sabina; Degorce, Sébastien; Fitzek, Martina; Green, Stephen; Hancox, Urs; Lambert-van der Brempt, Christine; Lohmann, Jean-Jacques; Maudet, Mickaël; Morgentin, Rémy; Péru, Aurélien; Plé, Patrick; Saleh, Twana; Ward, Lara; Warin, Nicolas Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 9(2016) Page Start: 2318 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗