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Author/Creator Fearon, Daren

1. An automatic pipeline for the design of irreversible derivatives identifies a potent SARS-CoV-2 Mpro inhibitor. Issue 12 (16th December 2021)

Authors:
Zaidman, Daniel; Gehrtz, Paul; Filep, Mihajlo; Fearon, Daren; Gabizon, Ronen; Douangamath, Alice; Prilusky, Jaime; Duberstein, Shirly; Cohen, Galit; Owen, C. David; Resnick, Efrat; Strain-Damerell, Claire; Lukacik, Petra; Barr, Haim; Walsh, Martin A.; von Delft, Frank; London, Nir
Journal:
Cell chemical biology
Issue:
Volume 28:Issue 12(2021)
Page Start:
1795
Record Type:
Journal Article
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2. Discovery of novel druggable pockets on polyomavirus VP1 through crystallographic fragment-based screening to develop capsid assembly inhibitors. Issue 8 (5th May 2022)

Authors:
Osipov, Evgenii M.; Munawar, Ali H.; Beelen, Steven; Fearon, Daren; Douangamath, Alice; Wild, Conor; Weeks, Stephen D.; Van Aerschot, Arthur; von Delft, Frank; Strelkov, Sergei V.
Journal:
RSC chemical biology
Issue:
Volume 3:Issue 8(2022)
Page Start:
1013
Record Type:
Journal Article
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3. Expanding the Repertoire of Low‐Molecular‐Weight Pentafluorosulfanyl‐Substituted Scaffolds. (22nd February 2022)

Authors:
Jose, Arathy; Guest, Daniel; LeGay, Remi; Tizzard, Graham J.; Coles, Simon J.; Derveni, Mariliza; Wright, Edward; Marrison, Lester; Lee, Alpha A.; Morris, Aaron; Robinson, Matt; von Delft, Frank; Fearon, Daren; Koekemoer, Lizbé; Matviuk, Tetiana; Aimon, Anthony; Schofield, Christopher J.; Malla, ...
Journal:
ChemMedChem
Issue:
Volume 17:Number 7(2022)
Page Start:
n/a
Record Type:
Journal Article
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4. Synthesis and profiling of a 3-aminopyridin-2-one-based kinase targeted fragment library: Identification of 3-amino-5-(pyridin-4-yl)pyridin-2(1H)-one scaffold for monopolar spindle 1 (MPS1) and Aurora kinases inhibition. Issue 11 (15th July 2018)

Authors:
Fearon, Daren; Westwood, Isaac M.; van Montfort, Rob L.M.; Bayliss, Richard; Jones, Keith; Bavetsias, Vassilios
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 26:Issue 11(2018)
Page Start:
3021
Record Type:
Journal Article
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