1. Discovery and Characterization of CD12681, a Potent RORγ Inverse Agonist, Preclinical Candidate for the Topical Treatment of Psoriasis. (6th February 2018) Authors: Ouvry, Gilles; Atrux‐Tallau, Nicolas; Bihl, Franck; Bondu, Aline; Bouix‐Peter, Claire; Carlavan, Isabelle; Christin, Olivier; Cuadrado, Marie‐Josée; Defoin‐Platel, Claire; Deret, Sophie; Duvert, Denis; Feret, Christophe; Forissier, Mathieu; Fournier, Jean‐François; Froude, David; Hacini‐Rachinel,... Journal: ChemMedChem Issue: Volume 13:Number 4(2018) Page Start: 321 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery and process development of a novel TACE inhibitor for the topical treatment of psoriasis. Issue 4 (15th February 2018) Authors: Boiteau, Jean-Guy; Ouvry, Gilles; Arlabosse, Jean-Marie; Astri, Stéphanie; Beillard, Audrey; Bhurruth-Alcor, Yushma; Bonnary, Laetitia; Bouix-Peter, Claire; Bouquet, Karine; Bourotte, Marilyne; Cardinaud, Isabelle; Comino, Catherine; Deprez, Benoît; Duvert, Denis; Féret, Angélique; Hacini-Rachine... Journal: Bioorganic & medicinal chemistry Issue: Volume 26:Issue 4(2018) Page Start: 945 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of phenoxyindazoles and phenylthioindazoles as RORγ inverse agonists. Issue 23 (1st December 2016) Authors: Ouvry, Gilles; Bouix-Peter, Claire; Ciesielski, Fabrice; Chantalat, Laurent; Christin, Olivier; Comino, Catherine; Duvert, Denis; Feret, Christophe; Harris, Craig S.; Lamy, Laurent; Luzy, Anne-Pascale; Musicki, Branislav; Orfila, Danielle; Pascau, Jonathan; Parnet, Véronique; Perrin, Agnès; Pierr... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 26:Issue 23(2016) Page Start: 5802 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Identification of novel TACE inhibitors compatible with topical application. Issue 8 (15th April 2017) Authors: Ouvry, Gilles; Berton, Yaël; Bhurruth-Alcor, Yushma; Bonnary, Laetitia; Bouix-Peter, Claire; Bouquet, Karine; Bourotte, Marilyne; Chambon, Sandrine; Comino, Catherine; Deprez, Benoît; Duvert, Denis; Duvert, Gwenaëlle; Hacini-Rachinel, Feriel; Harris, Craig S.; Luzy, Anne-Pascale; Mathieu, Arnaud;... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 8(2017) Page Start: 1848 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗