1. Discovery of a novel azetidine scaffold for colony stimulating factor-1 receptor (CSF-1R) Type II inhibitors by the use of docking models. Issue 1 (1st January 2019) Authors: Ikegashira, Kazutaka; Ikenogami, Taku; Yamasaki, Takayuki; Hase, Yasunori; Yamaguchi, Takayuki; Inagaki, Koji; Doi, Satoki; Adachi, Tsuyoshi; Koga, Yoshihisa; Hashimoto, Hiromasa Journal: Bioorganic & medicinal chemistry letters Issue: Volume 29:Issue 1(2019) Page Start: 115 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Fragment-based lead discovery to identify novel inhibitors that target the ATP binding site of pyruvate dehydrogenase kinases. (15th August 2021) Authors: Akaki, Tatsuo; Bessho, Yuki; Ito, Takashi; Fujioka, Shingo; Ubukata, Minoru; Mori, Genki; Yamanaka, Kenji; Orita, Takuya; Doi, Satoki; Iwanaga, Tomoko; Ikegashira, Kazutaka; Hantani, Yoshiji; Nakanishi, Isao; Adachi, Tsuyoshi Journal: Bioorganic & medicinal chemistry Issue: Volume 44(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Structure-based drug design of novel and highly potent pyruvate dehydrogenase kinase inhibitors. (15th December 2021) Authors: Bessho, Yuki; Akaki, Tatsuo; Hara, Yoshinori; Yamakawa, Maki; Obika, Shingo; Mori, Genki; Ubukata, Minoru; Yasue, Katsutaka; Nakane, Yoshitomi; Terasako, Yasuo; Orita, Takuya; Doi, Satoki; Iwanaga, Tomoko; Fujishima, Ayumi; Adachi, Tsuyoshi; Ueno, Hiroshi; Motomura, Takahisa Journal: Bioorganic & medicinal chemistry Issue: Volume 52(2021) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Ternary complex of human RORγ ligand‐binding domain, inverse agonist and SMRT peptide shows a unique mechanism of corepressor recruitment. (11th May 2017) Authors: Noguchi, Masato; Nomura, Akihiro; Murase, Ken; Doi, Satoki; Yamaguchi, Keishi; Hirata, Kazuyuki; Shiozaki, Makoto; Hirashima, Shintaro; Kotoku, Masayuki; Yamaguchi, Takayuki; Katsuda, Yoshiaki; Steensma, Ruo; Li, Xioalin; Tao, Haiyan; Tse, Bruno; Fenn, Morgan; Babine, Robert; Bradley, Erin; Crowe... Journal: Genes to cells Issue: Volume 22:Number 6(2017) Page Start: 535 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Ternary crystal structure of human RORγ ligand-binding-domain, an inhibitor and corepressor peptide provides a new insight into corepressor interaction. Issue 1 (December 2018) Authors: Noguchi, Masato; Nomura, Akihiro; Doi, Satoki; Yamaguchi, Keishi; Hirata, Kazuyuki; Shiozaki, Makoto; Maeda, Katsuya; Hirashima, Shintaro; Kotoku, Masayuki; Yamaguchi, Takayuki; Katsuda, Yoshiaki; Crowe, Paul; Tao, Haiyan; Thacher, Scott; Adachi, Tsuyoshi Journal: Scientific reports Issue: Volume 8:Issue 1(2018) Page Start: 1 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. The discovery of 3, 3-dimethyl-1, 2, 3, 4-tetrahydroquinoxaline-1-carboxamides as AMPD2 inhibitors with a novel mechanism of action. (15th January 2023) Authors: Kitao, Yuki; Saito, Tadataka; Watanabe, Satoshi; Ohe, Yasuhiro; Takahashi, Koichi; Akaki, Tatsuo; Adachi, Tsuyoshi; Doi, Satoki; Yamanaka, Kenji; Murai, Yasutaka; Oba, Makoto; Suzuki, Takayoshi Journal: Bioorganic & medicinal chemistry letters Issue: Volume 80(2023) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗