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Author/Creator Dabros, Marta

1. Discovery and SAR of aryl hydroxy pyrimidinones as potent small molecule agonists of the GPCR APJ. Issue 7 (1st April 2020)

Authors:
Myers, Michael C.; Bilder, Donna M.; Cavallaro, Cullen L.; Chao, Hannguang J.; Su, Shun; Burford, Neil T.; Nayeem, Akbar; Wang, Tao; Yan, Mujing; Langish, Robert A.; Dabros, Marta; Li, Yi-Xin; Rose, Anne V.; Behnia, Kamelia; Onorato, Joelle M.; Gargalovic, Peter S.; Wexler, Ruth R.; Lawrence, R. ...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 7(2020)
Page Start:
Record Type:
Journal Article
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2. Identification of bicyclic hexafluoroisopropyl alcohol sulfonamides as retinoic acid receptor-related orphan receptor gamma (RORγ/RORc) inverse agonists. Employing structure-based drug design to improve pregnane X receptor (PXR) selectivity. Issue 2 (15th January 2018)

Authors:
Gong, Hua; Weinstein, David S.; Lu, Zhonghui; Duan, James J.-W.; Stachura, Sylwia; Haque, Lauren; Karmakar, Ananta; Hemagiri, Hemalatha; Raut, Dhanya Kumar; Gupta, Arun Kumar; Khan, Javed; Camac, Dan; Sack, John S.; Pudzianowski, Andrew; Wu, Dauh-Rurng; Yarde, Melissa; Shen, Ding-Ren; Borowski, V...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 2(2018)
Page Start:
85
Record Type:
Journal Article
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3. Identification of potent tricyclic prodrug S1P1 receptor modulators12. Issue 4 (1st December 2016)

Authors:
Marcoux, David; Xiao, Hai-Yun; Murali Dhar, T. G.; Xie, Jenny; Lehman-McKeeman, Lois D.; Wu, Dauh-Rurng; Dabros, Marta; Yang, Xiaoxia; Taylor, Tracy L.; Zhou, Xia D.; Heimrich, Elizabeth M.; Thomas, Rochelle; McIntyre, Kim W.; Shi, Hong; Levesque, Paul C.; Sun, Huadong; Yang, Zheng; Marino, Antho...
Journal:
MedChemComm
Issue:
Volume 8:Issue 4(2017)
Page Start:
725
Record Type:
Journal Article
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