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- Crawforth, James [remove] 1
- 615.19 1
- ADMET absorption, distribution, metabolism, excretion and toxicity -- AUC area under the concentration versus time curve -- Clp plasma clearance -- Clu unbound clearance -- F bioavailability -- HLM human liver microsomes -- hERG human ether–a–go–go -- hHeps human hepatocytes -- IC50 half-maximum inhibitory concentration -- PK pharmacokinetics -- PMC parallel medicinal chemistry -- RRCK Ralph Russ canine kidney cell line -- T1/2 half-life -- TPSA topological surface area -- Vd volume of distribution 1
- Benzimidazole -- PF-06305591 -- Neuropathic pain -- Inflammatory pain -- Voltage gated sodium channel -- NaV1.8 -- SCN10A 1
- Biochemistry -- Periodicals 1
- Bioorganic chemistry -- Periodicals 1
- Chemistry, Clinical -- Periodicals 1
- Chemistry, Organic -- Periodicals 1
- Chimie bio-organique -- Périodiques 1
- Chimie pharmaceutique -- Périodiques 1
- Pharmaceutical chemistry -- Periodicals 1