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Author/Creator Conlon, Patrick

1. Optimization of novel reversible Bruton's tyrosine kinase inhibitors identified using Tethering-fragment-based screens. Issue 13 (1st July 2019)

Authors:
Hopkins, Brian T.; Bame, Eris; Bell, Noah; Bohnert, Tonika; Bowden-Verhoek, Jon K.; Bui, Minna; Cancilla, Mark T.; Conlon, Patrick; Cullen, Patrick; Erlanson, Daniel A.; Fan, Junfa; Fuchs-Knotts, Tarra; Hansen, Stig; Heumann, Stacey; Jenkins, Tracy J.; Marcotte, Douglas; McDowell, Bob; Mertsching...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 27:Issue 13(2019)
Page Start:
2905
Record Type:
Journal Article
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2. Utilizing structure based drug design and metabolic soft spot identification to optimize the in vitro potency and in vivo pharmacokinetic properties leading to the discovery of novel reversible Bruton's tyrosine kinase inhibitors. (15th August 2021)

Authors:
Hopkins, Brian T.; Bame, Eris; Bell, Noah; Bohnert, Tonika; Bowden-Verhoek, Jon K.; Bui, Minna; Cancilla, Mark T.; Conlon, Patrick; Cullen, Patrick; Erlanson, Daniel A.; Fan, Junfa; Fuchs-Knotts, Tarra; Hansen, Stig; Heumann, Stacey; Jenkins, Tracy J.; Gua, Chuck; Liu, Ying; Liu, YuTing; Lulla, M...
Journal:
Bioorganic & medicinal chemistry
Issue:
Volume 44(2021)
Page Start:
Record Type:
Journal Article
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3. Discovery of structural diverse reversible BTK inhibitors utilized to develop a novel in vivo CD69 and CD86 PK/PD mouse model. (15th January 2023)

Authors:
Vandeveer, George H.; Arduini, Robert M.; Baker, Darren P.; Barry, Kevin; Bohnert, Tonika; Bowden-Verhoek, Jon K.; Conlon, Patrick; Cullen, Patrick F.; Guan, Bing; Jenkins, Tracy J.; Liao, Shu-Yu; Lin, Lin; Liu, Yu-Ting; Marcotte, Douglas; Mertsching, Elisabeth; Metrick, Claire M.; Negrou, Ella; ...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 80(2023)
Page Start:
Record Type:
Journal Article
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