1. 2-Aminomethylthieno[3, 2-d]pyrimidin-4(3H)-ones bearing 3-methylpyrazole hinge binding moiety: Highly potent, selective, and time-dependent inhibitors of Cdc7 kinase. Issue 14 (15th July 2017) Authors: Kurasawa, Osamu; Homma, Misaki; Oguro, Yuya; Miyazaki, Tohru; Mori, Kouji; Uchiyama, Noriko; Iwai, Kenichi; Ohashi, Akihiro; Hara, Hideto; Yoshida, Sei; Cho, Nobuo Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 14(2017) Page Start: 3658 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Development of a degrader against oncogenic fusion protein FGFR3-TACC3. (15th March 2022) Authors: Shibata, Norihito; Cho, Nobuo; Koyama, Hiroo; Naito, Mikihiko Journal: Bioorganic & medicinal chemistry letters Issue: Volume 60(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Development of protein degradation inducers of oncogenic BCR‐ABL protein by conjugation of ABL kinase inhibitors and IAP ligands. Issue 8 (19th June 2017) Authors: Shibata, Norihito; Miyamoto, Naoki; Nagai, Katsunori; Shimokawa, Kenichiro; Sameshima, Tomoya; Ohoka, Nobumichi; Hattori, Takayuki; Imaeda, Yasuhiro; Nara, Hiroshi; Cho, Nobuo; Naito, Mikihiko Journal: Cancer science Issue: Volume 108:Issue 8(2017) Page Start: 1657 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Direct and practical synthesis of 2′-O, 4′-C-aminomethylene-bridged nucleic acid purine derivatives by transglycosylation. Issue 9 (2nd March 2017) Authors: Umemoto, Tadashi; Masada, Shinichi; Miyata, Kenichi; Ogasawara-Shimizu, Mari; Murata, Shumpei; Nishi, Kazunori; Ogi, Kazuhiro; Hayase, Yoji; Cho, Nobuo Journal: Tetrahedron Issue: Volume 73:Issue 9(2017) Page Start: 1211 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
5. Discovery of phenylpyrrolidine derivatives as a novel class of retinol binding protein 4 (RBP4) reducers. (15th January 2022) Authors: Nakamura, Shinji; Kamaura, Masahiro; Akao, Yuichiro; Nakamura, Natsuko; Mizukami, Atsushi; Goto, Akihiko; Furuyama, Naoki; Cho, Nobuo; Kasai, Shizuo Journal: Bioorganic & medicinal chemistry Issue: Volume 54(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
6. Identification of a new class of potent Cdc7 inhibitors designed by putative pharmacophore model: Synthesis and biological evaluation of 2, 3-dihydrothieno[3, 2-d]pyrimidin-4(1H)-ones. Issue 7 (1st April 2017) Authors: Kurasawa, Osamu; Oguro, Yuya; Miyazaki, Tohru; Homma, Misaki; Mori, Kouji; Iwai, Kenichi; Hara, Hideto; Skene, Robert; Hoffman, Isaac; Ohashi, Akihiro; Yoshida, Sei; Ishikawa, Tomoyasu; Cho, Nobuo Journal: Bioorganic & medicinal chemistry Issue: Volume 25:Issue 7(2017) Page Start: 2133 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
7. New antimalarials identified by a cell-based phenotypic approach: Structure–activity relationships of 2, 3, 4, 9-tetrahydro-1H-β-carboline derivatives possessing a 2-((coumarin-5-yl)oxy)alkanoyl moiety. (15th July 2022) Authors: Cho, Nobuo; Kikuzato, Ko; Futamura, Yushi; Shimizu, Takeshi; Hayase, Hiroki; Kamisaka, Kikuko; Takaya, Daisuke; Yuki, Hitomi; Honma, Teruki; Niikura, Mamoru; Kobayashi, Fumie; Watanabe, Nobumoto; Osada, Hiroyuki; Koyama, Hiroo Journal: Bioorganic & medicinal chemistry Issue: Volume 66(2022) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
8. SNIPER(TACC3) induces cytoplasmic vacuolization and sensitizes cancer cells to Bortezomib. Issue 5 (26th April 2017) Authors: Ohoka, Nobumichi; Nagai, Katsunori; Shibata, Norihito; Hattori, Takayuki; Nara, Hiroshi; Cho, Nobuo; Naito, Mikihiko Journal: Cancer science Issue: Volume 108:Issue 5(2017) Page Start: 1032 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗