1. Discovery of 7-(3-(piperazin-1-yl)phenyl)pyrrolo[2, 1-f][1, 2, 4]triazin-4-amine derivatives as highly potent and selective PI3Kδ inhibitors. Issue 4 (15th February 2017) Authors: Qin, Lan-Ying; Ruan, Zheming; Cherney, Robert J.; Dhar, T.G. Murali; Neels, James; Weigelt, Carolyn A.; Sack, John S.; Srivastava, Anurag S.; Cornelius, Lyndon A.M.; Tino, Joseph A.; Stefanski, Kevin; Gu, Xiaomei; Xie, Jenny; Susulic, Vojkan; Yang, Xiaoxia; Yarde-Chinn, Melissa; Skala, Stacey; Bo... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 4(2017) Page Start: 855 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Tricyclic sulfones as potent, selective and efficacious RORγt inverse agonists – Exploring C6 and C8 SAR using late-stage functionalization. Issue 23 (1st December 2020) Authors: Shi, Qing; Xiao, Zili; Yang, Michael G.; Marcoux, David; Cherney, Robert J.; Yip, Shiuhang; Li, Peng; Wu, Dauh-Rurng; Weigelt, Carolyn A.; Sack, John; Khan, Javed; Ruzanov, Max; Wang, Jinhong; Yarde, Melissa; Ellen Cvijic, Mary; Li, Sha; Shuster, David J.; Xie, Jenny; Sherry, Tara; Obermeier, Mary Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 23(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗