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Author/Creator Capstick, Rory A.

1. Discovery of a potent M5 antagonist with improved clearance profile. Part 1: Piperidine amide-based antagonists. (15th November 2022)

Authors:
Capstick, Rory A.; Whomble, David; Orsi, Douglas L.; Felts, Andrew S.; Rodriguez, Alice L.; Vinson, Paige N.; Chang, Sichen; Blobaum, Anna L.; Niswender, Colleen M.; Conn, P. Jeffrey; Jones, Carrie K.; Lindsley, Craig W.; Han, Changho
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 76(2022)
Page Start:
Record Type:
Journal Article
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2. Discovery of structurally distinct tricyclic M4 positive allosteric modulator (PAM) chemotypes – Part 2. (1st December 2021)

Authors:
Long, Madeline F.; Capstick, Rory A.; Spearing, Paul K.; Engers, Julie L.; Gregro, Alison R.; Bollinger, Sean R.; Chang, Sichen; Luscombe, Vincent B.; Rodriguez, Alice L.; Cho, Hyekyung P.; Niswender, Colleen M.; Bridges, Thomas M.; Conn, P. Jeffrey; Lindsley, Craig W.; Engers, Darren W.; Temple,...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 53(2021)
Page Start:
Record Type:
Journal Article
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Available online (eLD content is only available in our Reading Rooms) ↗

3. The discovery of VU0652957 (VU2957, Valiglurax): SAR and DMPK challenges en route to an mGlu4 PAM development candidate. Issue 2 (15th January 2019)

Authors:
Panarese, Joseph D.; Engers, Darren W.; Wu, Yong-Jin; Guernon, Jason M.; Chun, Aspen; Gregro, Alison R.; Bender, Aaron M.; Capstick, Rory A.; Wieting, Joshua M.; Bronson, Joanne J.; Macor, John E.; Westphal, Ryan; Soars, Matthew; Engers, Julie E.; Felts, Andrew S.; Rodriguez, Alice L.; Emmitte, K...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 29:Issue 2(2019)
Page Start:
342
Record Type:
Journal Article
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Available online (eLD content is only available in our Reading Rooms) ↗

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