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Author/Creator Bollinger, Sean R.

1. Discovery and characterization of N-(1, 3-dialkyl-1H-indazol-6-yl)-1H-pyrazolo[4, 3-b]pyridin-3-amine scaffold as mGlu4 positive allosteric modulators that mitigate CYP1A2 induction liability. Issue 15 (15th August 2018)

Authors:
Engers, Darren W.; Bollinger, Sean R.; Engers, Julie L.; Panarese, Joseph D.; Breiner, Megan M.; Gregro, Alison; Blobaum, Anna L.; Bronson, Joanne J.; Wu, Yong-Jin; Macor, John E.; Rodriguez, Alice L.; Zamorano, Rocio; Conn, P. Jeffrey; Lindsley, Craig W.; Niswender, Colleen M.; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 28:Issue 15(2018)
Page Start:
2641
Record Type:
Journal Article
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2. Discovery of structurally distinct tricyclic M4 positive allosteric modulator (PAM) chemotypes – Part 2. (1st December 2021)

Authors:
Long, Madeline F.; Capstick, Rory A.; Spearing, Paul K.; Engers, Julie L.; Gregro, Alison R.; Bollinger, Sean R.; Chang, Sichen; Luscombe, Vincent B.; Rodriguez, Alice L.; Cho, Hyekyung P.; Niswender, Colleen M.; Bridges, Thomas M.; Conn, P. Jeffrey; Lindsley, Craig W.; Engers, Darren W.; Temple,...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 53(2021)
Page Start:
Record Type:
Journal Article
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3. Discovery, synthesis and characterization of a series of 7-aryl-imidazo[1, 2-a]pyridine-3-ylquinolines as activin-like kinase (ALK) inhibitors. Issue 18 (15th September 2020)

Authors:
Engers, Darren W.; Bollinger, Sean R.; Felts, Andrew S.; Vadukoot, Anish K.; Williams, Charles H.; Blobaum, Anna L.; Lindsley, Craig W.; Hong, Charles C.; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 30:Issue 18(2020)
Page Start:
Record Type:
Journal Article
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4. Synthesis and structure–activity relationships of a series of 4-methoxy-3-(piperidin-4-yl)oxy benzamides as novel inhibitors of the presynaptic choline transporter. Issue 8 (15th April 2015)

Authors:
Bollinger, Sean R.; Engers, Darren W.; Ennis, Elizabeth A.; Wright, Jane; Locuson, Charles W.; Lindsley, Craig W.; Blakely, Randy D.; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 8(2015)
Page Start:
1757
Record Type:
Journal Article
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5. Synthesis and structure–activity relationships of a series of 4-methoxy-3-(piperidin-4-yl)oxy benzamides as novel inhibitors of the presynaptic choline transporter. Issue 8 (15th April 2015)

Authors:
Bollinger, Sean R.; Engers, Darren W.; Ennis, Elizabeth A.; Wright, Jane; Locuson, Charles W.; Lindsley, Craig W.; Blakely, Randy D.; Hopkins, Corey R.
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 25:Issue 8(2015)
Page Start:
1757
Record Type:
Journal Article
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Available online (eLD content is only available in our Reading Rooms) ↗

6. VU6005806/AZN-00016130, an advanced M4 positive allosteric modulator (PAM) profiled as a potential preclinical development candidate. Issue 14 (15th July 2019)

Authors:
Engers, Darren W.; Melancon, Bruce J.; Gregro, Allison R.; Bertron, Jeanette L.; Bollinger, Sean R.; Felts, Andrew S.; Konkol, Leah C.; Wood, Michael R.; Bollinger, Katrina A.; Luscombe, Vincent B.; Rodriguez, Alice L.; Jones, Carrie K.; Bubser, Michael; Yohn, Samantha E.; Wood, Michael W.; Brand...
Journal:
Bioorganic & medicinal chemistry letters
Issue:
Volume 29:Issue 14(2019)
Page Start:
1714
Record Type:
Journal Article
View Content:
Available online (eLD content is only available in our Reading Rooms) ↗