1. Discovery of 1H-pyrazolo[3, 4-b]pyridines as potent dual orexin receptor antagonists (DORAs). Issue 23 (1st December 2015) Authors: Behnke, Dirk; Cotesta, Simona; Hintermann, Samuel; Fendt, Markus; Gee, Christine E.; Jacobson, Laura H.; Laue, Grit; Meyer, Arndt; Wagner, Trixie; Badiger, Sangamesh; Chaudhari, Vinod; Chebrolu, Murali; Pandit, Chetan; Hoyer, Daniel; Betschart, Claudia Journal: Bioorganic & medicinal chemistry letters Issue: Volume 25:Issue 23(2015) Page Start: 5555 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of potent, orally bioavailable in vivo efficacious antagonists of the TLR7/8 pathway. Issue 17 (1st September 2020) Authors: Alper, Phil B.; Deane, Jonathan; Betschart, Claudia; Buffet, David; Collignon Zipfel, Géraldine; Gordon, Perry; Hampton, Janice; Hawtin, Stuart; Ibanez, Maureen; Jiang, Tao; Junt, Tobias; Knoepfel, Thomas; Liu, Bo; Maginnis, Jillian; McKeever, Una; Michellys, Pierre-Yves; Mutnick, Daniel; Nayak, ... Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 17(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗