1. Discovery of N-substituted 7-azaindoles as Pan-PIM kinase inhibitors – Lead series identification – Part II. Issue 20 (15th October 2017) Authors: Barberis, Claude; Moorcroft, Neil; Pribish, James; Tserlin, Elina; Gross, Alexandre; Czekaj, Mark; Barrague, Matthieu; Erdman, Paul; Majid, Tahir; Batchelor, Joseph; Levit, Mikhail; Hebert, Andrew; Shen, Liduo; Moreno-Mazza, Sandra; Wang, Anlai Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 20(2017) Page Start: 4735 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
2. Discovery of N-substituted 7-azaindoles as Pan-PIM kinases inhibitors – Lead optimization – Part III. Issue 3 (1st February 2019) Authors: Barberis, Claude; Pribish, James; Tserlin, Elina; Gross, Alexandre; Czekaj, Mark; Barragué, Matthieu; Erdman, Paul; Maniar, Sachin; Jiang, John; Fire, Luke; Patel, Vinod; Hebert, Andrew; Levit, Mikhail; Wang, Anlai; Sun, Frank; Huang, Shih-Min A. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 29:Issue 3(2019) Page Start: 491 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
3. Discovery of N-substituted 7-azaindoles as PIM1 kinase inhibitors – Part I. Issue 20 (15th October 2017) Authors: Barberis, Claude; Moorcroft, Neil; Arendt, Chris; Levit, Mikhail; Moreno-Mazza, Sandra; Batchelor, Joseph; Mechin, Ingrid; Majid, Tahir Journal: Bioorganic & medicinal chemistry letters Issue: Volume 27:Issue 20(2017) Page Start: 4730 Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗
4. Discovery of SARxxxx92, a pan-PIM kinase inhibitor, efficacious in a KG1 tumor model. Issue 23 (1st December 2020) Authors: Barberis, Claude; Erdman, Paul; Czekaj, Mark; Fire, Luke; Pribish, James; Tserlin, Elina; Maniar, Sachin; Batchelor, Joseph D.; Liu, Jinyu; Patel, Vinod F.; Hebert, Andrew; Levit, Mikhail; Wang, Anlai; Sun, Frank; Huang, Shih-Min A. Journal: Bioorganic & medicinal chemistry letters Issue: Volume 30:Issue 23(2020) Page Start: Record Type: Journal Article View Content: Available online (eLD content is only available in our Reading Rooms) ↗